Target Details
UniProt ACP08912
Gene SymbolCHRM5
Protein NameMuscarinic acetylcholine receptor M5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 585
  • Clinical molecules 27
  • Avg pChEMBL 7.09
Top Co-occurrence Targets
Active Molecules (585)
InChIKey pChEMBL Type Targets Clinical
WTRLYZUEDFZGKI 8.6 Ki 5
BNLVIXOVYRJUTA 8.6 Ki 5
UOKGNINOAYOIDX 8.6 Ki 5
JGOIBENTSQHWDQ 8.6 Ki 5
XUENORREMLOMPD 8.6 Ki 5
NCPVINAZNPBCKE 8.6 Ki 5
PFSPMYHTZUFJQW 8.5 Ki 5
VPWKHNIBDCHPNN 8.5 Ki 5
QCUQACXEVHRHIF 8.5 Ki 5
JJCFRYNCJDLXIK 8.5 IC50 25 Yes
UJXAGMVNACHDOG 8.5 Ki 5
WCMVSMOIDILBOJ 8.5 Ki 5
MVNBPMNELMRFMU 8.5 Ki 5
NEQYHZCZFMESJN 8.5 Ki 5
AFLBGAQHDSOPKA 8.5 Ki 5
PCEDEEWEONTUHP 8.4 Kd 5
ZRYHPQCHHOKSMD 8.4 Ki 4
UFSZYKLBZJNXLV 8.4 Ki 5
INEDRTXKDAPQKU 8.4 Ki 5
KKEGQSSUXOGEAF 8.4 Ki 5
STECJAGHUSJQJN 8.3 Ki 5
QZQDZBWQUNVCFF 8.3 Ki 5
VPJXQGSRWJZDOB 8.3 Ki 7
ROEXPZFFOZZHOY 8.3 Ki 5
OANBYDFPBWKVGI 8.3 Ki 5
PCEDEEWEONTUHP 8.3 Kd 5
BMNOFIWIZFZYES 8.3 Ki 5
UKDFFUWYVUWORH 8.3 Ki 2
FZXSXMYFIZKXPT 8.2 Ki 12
JOMFXRAREZYSMG 8.2 Ki 5
UJXAGMVNACHDOG 8.2 Ki 5
WOMCGBFNBSIIEA 8.2 Kd 5
CJGNMVAAMQAWEF 8.2 Ki 16
OYYDSUSKLWTMMQ 8.2 Ki 5
TYLFZULSDOOCRC 8.2 Ki 5
DCNMFOFKZLIEDY 8.2 Ki 5
MAGHIFWNWZHPQG 8.2 Ki 5
YSXKPIUOCJLQIE 8.2 Ki 5
XIQVNETUBQGFHX 8.2 Ki 10
MMUOGZOUFNQXMP 8.2 Ki 5
MVNBPMNELMRFMU 8.2 Ki 5
IPPGGAXXAKWHHQ 8.1 Ki 5
UECHFIXSINCEDW 8.1 Ki 5
MLPXDKWFNNRLJM 8.1 Ki 4
KLBQZWRITKRQQV 8.1 IC50 25 Yes
PULJCGFLKSMODH 8.1 Ki 5
QQPVAVCRPBYZDM 8.1 IC50 2
NEUSVAOJNUQRTM 8.1 IC50 13 Yes
SQVWTVHVWIHOSU 8.1 Ki 5
UACRHRRJJCXGPC 8.0 Ki 5
2D structure