Target Details
| UniProt AC | P08912 |
|---|---|
| Gene Symbol | CHRM5 |
| Protein Name | Muscarinic acetylcholine receptor M5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 585
- Clinical molecules 27
- Avg pChEMBL 7.09
KEGG Pathways (7)
Active Molecules (585)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ORKIMQYINJNMRH
|
6.1 | Ki | 2 | — | |
QGWIQIAWOCJRPI
|
6.1 | Ki | 6 | — | |
XAPDCGAVGSRGKC
|
6.1 | IC50 | 2 | — | |
AWEBVNCNTLOVSN
|
6.1 | Ki | 5 | — | |
OGAKLTJNUQRZJU
|
6.1 | Ki | 9 | — | |
PWYNNAYMPKVKJL
|
6.1 | Kd | 5 | — | |
RHAFROHARIZTPJ
|
6.1 | Kd | 5 | — | |
AVNRDCQRRUOTCC
|
6.1 | Ki | 4 | — | |
NGKTYFBTWFLIRS
|
6.1 | Ki | 4 | — | |
OPURXCGDAMNMQI
|
6.1 | Ki | 2 | — | |
QDGDDAFKQVQWCI
|
6.1 | Ki | 5 | — | |
UPDAFPDJKSGPME
|
6.1 | Ki | 5 | — | |
YZDFADGMVOSVIX
|
6.1 | Ki | 16 | — | |
ZPASGLGRGIEHTG
|
6.1 | IC50 | 2 | — | |
SBWDNXAOTCMVAA
|
6.0 | IC50 | 7 | — | |
LQOJFNRTYZDTBR
|
6.0 | Ki | 5 | — | |
MYQTVOSXIIRICR
|
6.0 | Ki | 5 | — | |
BHNWCPXBMCJVAS
|
6.0 | Ki | 5 | — | |
CWPKTBMRVATCBL
|
6.0 | Ki | 8 | — | |
PSBBAGWMKGXQRW
|
6.0 | Ki | 9 | — | |
RSDOPYMFZBJHRL
|
6.0 | Kd | 5 | — | |
SPHRJZBOFYIKMC
|
6.0 | Ki | 4 | — | |
UPPZIKNLEDOKKO
|
6.0 | Ki | 5 | — | |
WWXCWTRLUXMAHX
|
6.0 | Ki | 7 | — | |
KXGAHULLQRZYOM
|
6.0 | Ki | 5 | — | |
UFFHNEZNXKJHFB
|
6.0 | Ki | 10 | — | |
WEGLOYDTDILXDA
|
6.0 | Ki | 22 | — | |
WYWIFABBXFUGLM
|
6.0 | Ki | 17 | — | |
GIIZNNXWQWCKIB
|
6.0 | Ki | 10 | — | |
QCOZXCKWZLHYKC
|
6.0 | Ki | 4 | — | |
RTHCYVBBDHJXIQ
|
6.0 | Ki | 15 | — | |
VDRDKKLNMTZAMF
|
6.0 | Ki | 2 | — | |
WKWADEWWLCVVLF
|
6.0 | Ki | 14 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — | |
WXGLQWLONQSHMW
|
6.0 | Ki | 3 | — |