Target Details
UniProt ACP08912
Gene SymbolCHRM5
Protein NameMuscarinic acetylcholine receptor M5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 585
  • Clinical molecules 27
  • Avg pChEMBL 7.09
Top Co-occurrence Targets
Active Molecules (585)
InChIKey pChEMBL Type Targets Clinical
GXDALQBWZGODGZ 6.2 IC50 21 Yes
KLQQZEIBZUZRLW 6.2 Ki 4
VMWJMSDTGWMQGP 6.2 IC50 4
XRPVRNLTTMYYDS 6.2 Ki 5
AGVQGHLXLYNMSL 6.2 Ki 5
CTLCSFGCIVNYGV 6.2 Ki 5
WQWPUTDMTVRSDR 6.2 Kd 5
DMFXETUOWLUQID 6.2 Ki 5
HTYJHPPHBQRXGX 6.2 Ki 5
MLKITGHXXPWOSH 6.2 Ki 5
WIHMMKGUBDZGEG 6.2 IC50 7
XEDHVZKDSYZQBF 6.2 Ki 7
YEWCXJGTKBDZNL 6.2 Ki 2
DERZBLKQOCDDDZ 6.2 IC50 20 Yes
HWEGXFSUSOJEQJ 6.2 Ki 3
KZLOJWPPQXXGJS 6.2 Ki 5
LJVNYCDXBXGQIK 6.2 Ki 14 Yes
MTDYDDJVCIHZKH 6.2 Ki 7
RVQVUMIXBGFJLZ 6.2 Ki 7
NJWRXZDGANXMDC 6.2 Ki 5
RCPNNLKDMRCWCD 6.2 Ki 5
YFWMVRIRFFWDJL 6.2 Ki 5
OCOMTFATMRIOSP 6.2 IC50 5
CAGFDMXWWOBBHR 6.2 Ki 5
JKGARLBCOXRROD 6.2 Ki 5
KTMWGHBDOVXVOW 6.2 Ki 4
OBLWLENBNRYSCO 6.1 IC50 5
QWGDMFLQWFTERH 6.1 IC50 23 Yes
RPUXCIYWJSVFFV 6.1 Ki 6
SVJMLYUFVDMUHP 6.1 Ki 26
VICTYDRNEFPKTN 6.1 Ki 5
MWFQIDNMZVEVKH 6.1 Ki 2
SOYKEARSMXGVTM 6.1 Ki 8
MVMQESMQSYOVGV 6.1 Ki 6
NBAPIQQREIVGBA 6.1 Ki 5
OJINAULTAMERKJ 6.1 Ki 8
PAYAQSDGYIQGSL 6.1 Ki 2
ANUNMVJZPWGZDH 6.1 Ki 5
CYXKNKQEMFBLER 6.1 Ki 5
DDXKWKGIBLVYQU 6.1 Ki 5
CWSRXZGMHUIVTH 6.1 IC50 4
JRUSYSCSOBAJQG 6.1 Ki 5
MVMQESMQSYOVGV 6.1 Ki 6
OIPILFWXSMYKGL 6.1 Ki 6
SMANXXCATUTDDT 6.1 Ki 25 Yes
TWUZJTIHFYRNSV 6.1 Ki 3
YVENIGOVHPMTDH 6.1 Ki 23
UBGMVJXVELKNMU 6.1 Ki 5
XTDVAENSULGVTJ 6.1 Ki 5
BCUGCHZRMKTPMU 6.1 Ki 6
2D structure