Target Details
UniProt ACP08912
Gene SymbolCHRM5
Protein NameMuscarinic acetylcholine receptor M5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 585
  • Clinical molecules 27
  • Avg pChEMBL 7.09
Top Co-occurrence Targets
Active Molecules (585)
InChIKey pChEMBL Type Targets Clinical
VMJSEWCRPGCNOF 6.3 Ki 5
VSWYSDPXUHVQCG 6.3 Ki 11
HHDGJFBTFPNSEV 6.3 Ki 5
WEGLOYDTDILXDA 6.3 Ki 22
XBBANBCTQDQYBC 6.3 Ki 4
MZDYABXXPZNUCT 6.3 Ki 5
RYSPLPSTYIIBHP 6.3 IC50 3
UVKZSORBKUEBAZ 6.3 IC50 13 Yes
BZBLQCBDTFEROJ 6.3 Ki 3
COCYKMCRONGNER 6.3 Ki 3
CQYGJUKSNQPNJR 6.3 Ki 3
ILAZBCOZIJMNAN 6.3 Ki 5
INUAAAUHEVUAGY 6.3 Ki 3
KDDCYVRQXRCCPT 6.3 Ki 4
KKOOZXHGLNSYOQ 6.3 Ki 3
KQDLURQMDUCAFL 6.3 Ki 3
LXHDJDGOVRXFAY 6.3 Ki 2
MONFTSPGJAUKAQ 6.3 Ki 3
NNMHVNSZEZYWLQ 6.3 Ki 4
NQBTZXNQBCBXSM 6.3 Ki 3
OTRATODOMCPGQI 6.3 Ki 5
PFQNHVGTLFNXFJ 6.3 Ki 4
QLHPXZICVIHDES 6.3 Ki 4
RQJNIMUZOJATIT 6.3 Ki 3
RTNLSUYWOQRWMP 6.3 Ki 4
RXJJLNUPBMTGAW 6.3 Ki 5
RXJJLNUPBMTGAW 6.3 Ki 5
RXSNACAZEYSDGE 6.3 Ki 3
RXTGAWLNZFDKJO 6.3 Ki 2
SFSDXYWNODMHCY 6.3 Ki 5
TWEXWSGNHKGNHI 6.3 Ki 4
UCDAGGLRRYYIRU 6.3 Ki 3
UEUYDRJDYJUBTN 6.3 Ki 3
UPQFMOHGVPABFY 6.3 Ki 3
WFHGMWHPBQUAFQ 6.3 Ki 3
WTNHCZORDQEROL 6.3 Ki 4
YWBLUYIJHOWRBA 6.3 Ki 4
ZQYPSZMHKOQOEF 6.3 Ki 4
IPNOLIDZPPDWLV 6.2 IC50 4
QIXOXAUNCKVBGL 6.2 Ki 5
CBDJZHFJKQNGLM 6.2 Ki 5
FWVRMDGONFOSIW 6.2 Ki 5
HNQCDUJRXDPLHW 6.2 Ki 5
LCJWZLPNZLCYKB 6.2 Ki 5
LLBLNMUONVVVPG 6.2 Ki 17
RSMOYRFTQUYBTP 6.2 Ki 5
UECJYWWGFQYNFJ 6.2 Kd 5
PKERJUIAPINEEV 6.2 Ki 5
BJUQLFXRXSMDCM 6.2 Ki 5
CHZUEGVOEFMIJH 6.2 Ki 8
2D structure