Target Details
UniProt ACP08912
Gene SymbolCHRM5
Protein NameMuscarinic acetylcholine receptor M5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 585
  • Clinical molecules 27
  • Avg pChEMBL 7.09
Top Co-occurrence Targets
Active Molecules (585)
InChIKey pChEMBL Type Targets Clinical
LERNTVKEWCAPOY 10.3 IC50 5
UKXSKSHDVLQNKG 10.3 Ki 5
XXWOCVWJOICKHA 10.1 Kd 5
LERNTVKEWCAPOY 10.0 Ki 6
WCMVSMOIDILBOJ 10.0 Ki 5
WOMCGBFNBSIIEA 9.9 Ki 5
ASMXXROZKSBQIH 9.8 IC50 5
WGOJWDWKHJHXSV 9.8 Ki 5
ANGKOCUUWGHLCE 9.7 IC50 5
GWAMGWDJCYIREE 9.7 Kd 20
HGMITUYOCPPQLE 9.7 Ki 5
IWBMAAUPHUCYCI 9.7 Kd 20
MODBIBJHAWXYOZ 9.7 Kd 20
WCMVSMOIDILBOJ 9.7 Ki 5
ZRQMUCDHVVOENY 9.7 Kd 17
WOMCGBFNBSIIEA 9.6 Ki 5
LZCOQTDXKCNBEE 9.5 Ki 5
AFLBGAQHDSOPKA 9.4 Ki 5
HYJRTXSYDAFGJK 9.4 IC50 5
XXWOCVWJOICKHA 9.3 Kd 5
RKUNBYITZUJHSG 9.3 Ki 5
DVVFXQIXRYZXNS 9.3 Ki 5
RKUNBYITZUJHSG 9.2 Ki 5
QOXJSXPGWIRRNX 9.2 Ki 5
UFSZYKLBZJNXLV 9.2 Ki 5
WCMVSMOIDILBOJ 9.1 Ki 5
RKUNBYITZUJHSG 9.1 Ki 7
ZZCCWXNFFGHRJX 9.0 Ki 5
OEXHQOGQTVQTAT 9.0 Ki 5
OLYUOAVKDLVFLJ 9.0 Ki 5
UCURTLDVWIWPRM 8.9 Ki 5
DFCLHAWGKPEFIX 8.9 Ki 5
STECJAGHUSJQJN 8.9 Ki 4
OEXHQOGQTVQTAT 8.9 Ki 5
DFCLHAWGKPEFIX 8.9 Ki 5
UOKGNINOAYOIDX 8.8 Ki 5
AVNRDCQRRUOTCC 8.8 Ki 5
GIJXKZJWITVLHI 8.8 IC50 16
KKEGQSSUXOGEAF 8.8 Ki 5
NDXFHBBFUCQHAL 8.8 Ki 5
OANBYDFPBWKVGI 8.7 Ki 5
UBXUDWCOFMMEAI 8.7 Ki 5
CURUTKGFNZGFSE 8.7 IC50 10
DFCLHAWGKPEFIX 8.7 Ki 5
DFCLHAWGKPEFIX 8.7 Ki 5
LBOJYSIDWZQNJS 8.7 IC50 9
NPNXPJMTHYXCHW 8.7 Ki 4
AKMDZGUFAAEGFX 8.7 Ki 5
OOGJQPCLVADCPB 8.7 Ki 9
HXGBXQDTNZMWGS 8.6 Ki 8
2D structure