Target Details
UniProt ACP08908
Gene SymbolHTR1A
Protein Name5-hydroxytryptamine receptor 1A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 3,572
  • Clinical molecules 89
  • Avg pChEMBL 7.64
Top Co-occurrence Targets
Active Molecules (3,572)
InChIKey pChEMBL Type Targets Clinical
RKFRMULEVKBANT 9.0 Ki 3
ZZBUJMUPYXVJGM 9.0 Ki 2
IRNNHEZQBOQPHZ 9.0 Ki 4
BYHQOSOPNSLUAD 9.0 Ki 3
CZMNVXMBURYBAI 9.0 Ki 4
HFEAGUBAIYKXAC 9.0 Ki 2
XTICRBGKPDRHCR 9.0 Ki 4
AHJHJVULSVKBEA 9.0 Ki 5
ATIJQZLSMDZBIR 9.0 Ki 2
AYYCFGDXLUPJAQ 9.0 Ki 5
BCGWQEUPMDMJNV 9.0 IC50 30 Yes
CDQNHZRQGKLBDW 9.0 Ki 2
CGVZEZGEEUBAEK 9.0 Ki 3
DUKNIHFTDAXJON 9.0 Ki 13
IKINOGQZTQWAIL 9.0 Ki 3
IOKDDLUMOKQUEG 9.0 Ki 4
MZBZALUTJALVLT 9.0 Ki 4
NRFJXDLMBKNOHP 9.0 Ki 3
NSMCYUMPIGJKHV 9.0 Ki 9
PGMRWJOSCVZPRO 9.0 Ki 2
TYIREBTWRRZFOA 9.0 Ki 2
VAYOSLLFUXYJDT 9.0 Ki 19
VPCBUIFZQHYYDU 9.0 Ki 4
WAEVDDXBNJUJNE 9.0 Ki 8
WOHMWCGVHSYPFG 9.0 IC50 3
WRRJZZBXRRDBBD 9.0 IC50 3
YDPSNCPFCJTQRW 9.0 Ki 2
ZXGRMQACDGUTBN 9.0 Ki 4
IOFYRLZQZMPYGN 8.9 Ki 2
OHIHGZWNDVVIBE 8.9 Ki 2
WBENNDOANVTGAH 8.9 Ki 2
DSEPKSLFXGYPIU 8.9 IC50 3
IXXRJDPEMQTXTR 8.9 Ki 2
KWNJJPLLFRQMRI 8.9 Ki 4
LWBZBWXDCWJUBA 8.9 Ki 5
NLAPYFUIFIHYFO 8.9 Ki 3
NZGWRTVGHIZQDX 8.9 Ki 3
PLKOFQSGOPKBMP 8.9 Ki 3
PZZTZOMXZRXURK 8.9 Ki 2
UYZCRXKULSDXTA 8.9 Ki 4
VRRJFCMGNMFNOE 8.9 Ki 2
WALPSENJUDWNLI 8.9 Ki 2
DUUXVHJVUBCPDT 8.9 Ki 2
BHFRJLAPJAERKC 8.9 IC50 2
BMCUOUFSLYKUKP 8.9 Ki 3
DDSXQLHFTRQRQJ 8.9 Ki 3
GHBSODKXXQMXAV 8.9 Ki 3
GXMYCNTVOUYSEA 8.9 Ki 3
JESLIPCZKNHJMZ 8.9 Ki 2 Yes
KJVMAQQFBLAGOS 8.9 Ki 3
2D structure