Target Details
| UniProt AC | P08908 |
|---|---|
| Gene Symbol | HTR1A |
| Protein Name | 5-hydroxytryptamine receptor 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 3,572
- Clinical molecules 89
- Avg pChEMBL 7.64
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (3,572)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LLBLNMUONVVVPG
|
6.0 | Ki | 17 | — | |
NRYJUVLALBJESR
|
6.0 | Ki | 4 | — | |
NYBQQHJGLBCUBL
|
6.0 | Ki | 5 | — | |
OERJWHNFTHRHHI
|
6.0 | Ki | 3 | — | |
OOKNJSVAHXTYKL
|
6.0 | Ki | 3 | — | |
ORJIHHLJBCQRBS
|
6.0 | Ki | 6 | — | |
PCFGMPNKAUVMPL
|
6.0 | Ki | 2 | — | |
PHCCFIGNVNPMML
|
6.0 | IC50 | 7 | — | |
PXEURUZEVKVPGJ
|
6.0 | IC50 | 5 | — | |
QQJHRQZZCNYDMX
|
6.0 | Ki | 11 | — | |
SHOJVFLWKSRVPH
|
6.0 | Ki | 2 | — | |
UNRCJLILBVLZDQ
|
6.0 | Ki | 6 | — | |
UNRCJLILBVLZDQ
|
6.0 | Ki | 6 | — | |
VCFMMDVFGUQTHR
|
6.0 | Ki | 5 | — | |
VHGCDTVCOLNTBX
|
6.0 | Ki | 19 | — | |
VTQSIRZSABRYHH
|
6.0 | Ki | 3 | — | |
WCXYNCOEJKTKIB
|
6.0 | Ki | 3 | — | |
XYJTURUCNQJUDF
|
6.0 | Ki | 3 | — | |
YKUHLXRZNYUNSP
|
6.0 | Ki | 5 | — | |
YOGJZQGRTVMCPY
|
6.0 | IC50 | 17 | — | |
YVWGGGGMRDLOGA
|
6.0 | Ki | 2 | — | |
YWXWHMFUKATDEE
|
6.0 | Ki | 2 | — |