Target Details
UniProt ACP08908
Gene SymbolHTR1A
Protein Name5-hydroxytryptamine receptor 1A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 3,572
  • Clinical molecules 89
  • Avg pChEMBL 7.64
Top Co-occurrence Targets
Active Molecules (3,572)
InChIKey pChEMBL Type Targets Clinical
RTTBMUKLKYPQQK 6.1 Ki 4
XBHTWHZBPNLIOV 6.1 Ki 3
YYBRTGMBVYRIBV 6.1 Ki 3
ZRMFHWUDQQZCJM 6.1 Ki 4
ALDCLQHVTZPMQV 6.1 Ki 3
BETHXCLHMRGYBW 6.1 Ki 9 Yes
BETVPTZOBIULKH 6.1 Ki 2
CZOXEMUHIJZXSF 6.1 Ki 6
CZPHWPDUDLEVFW 6.1 Ki 2
JTENRKUQAXBDKF 6.1 Ki 5
MUFITXOADYQFSV 6.1 Ki 2
PYMZBBSVTWGBTF 6.1 Ki 4
QPPKZPPBKXTTNB 6.1 Ki 3
ADWCVCJMIQYGTM 6.1 Ki 2
CJAWPFJGFFNXQI 6.1 Kd 4
DCSUBABJRXZOMT 6.1 Ki 24
FPCCSQOGAWCVBH 6.1 Kd 16
GCIDJPAHOAQOPY 6.1 Ki 3
GZXNMNCAWGIAAW 6.1 Ki 7 Yes
MNYODQSAKDAGDY 6.1 Ki 3
NXCCMUDPNPXACY 6.1 Ki 2 Yes
OLAXNDRKNPEFSN 6.1 Ki 3
SHILVAMBAMVDBR 6.1 Ki 2
UFFHNEZNXKJHFB 6.1 Ki 10
WFMXGGGKNJIUGJ 6.1 Ki 5
WSPGJGOBUJGMBV 6.1 Ki 2 Yes
XIMFQVXENHJKEO 6.1 Ki 10
XIMFQVXENHJKEO 6.1 Ki 10
YASBOGFWAMXINH 6.1 Kd 4
YLPJQEDKFKCTSE 6.1 Ki 4
AKGAFPAMSJSPPN 6.1 Ki 2
BAIXKGAZCOGILC 6.1 Ki 3
BVYRODJRYHZDHU 6.1 Ki 2
DGWDNZHZPVHEAC 6.1 Ki 2
GWBXCMYQCTUKHM 6.1 Ki 2
JVNZVNCHIUVRJV 6.1 IC50 2
QTNMHOVGTBINTB 6.1 Ki 2
SGVJKODGLNRNLW 6.1 Ki 18
BUNPANXQBOTFPV 6.1 Ki 3
BZDGCBXVIKXHFH 6.1 IC50 7
HKRNYOZJJMFDBV 6.1 IC50 2
KMWKXYYYWRNCEV 6.1 Ki 3
MNZKMXOYJBDBSR 6.1 Ki 7
OQGAVEZMVJJWSH 6.1 Ki 4
PBMOMMUCOYVEFZ 6.1 Ki 2
UZRMRNOPEVQTSO 6.1 Ki 3
XBNNPPLRTCDVRJ 6.1 Ki 4
ZAGAUUVCYGSPBP 6.1 Ki 3
CTJRXEBAFHPXDV 6.1 Ki 4
JHVNSHBHMRPFIN 6.1 Ki 2
2D structure