Target Details
UniProt ACP08908
Gene SymbolHTR1A
Protein Name5-hydroxytryptamine receptor 1A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 3,572
  • Clinical molecules 89
  • Avg pChEMBL 7.64
Top Co-occurrence Targets
Active Molecules (3,572)
InChIKey pChEMBL Type Targets Clinical
ACKGCCXJFAZCFF 6.2 Ki 7
FBDANPRMCCLYRK 6.2 Ki 3
GOTMKOSCLKVOGG 6.2 Ki 9
HGHZRWWRCHMWQC 6.2 Ki 4
HPMRFMKYPGXPEP 6.2 Ki 10
MRYWDVLOYWQXCU 6.2 Ki 3
ODCAEXNEGXTNBY 6.2 Ki 6
REMMHZSMZDLMEO 6.2 IC50 2
RUGBLRYISYKONW 6.2 Ki 3
WPSIPVCJWLGMEF 6.2 Ki 2
XZPGIQSKRLUYSY 6.2 Ki 2
ZDPNKNSRWQOPMC 6.2 IC50 2
ZTBBOIYRZHAFIN 6.2 Ki 8
GDRLBCZDGQFDCZ 6.2 Ki 7
HAULDNLFSXGWJR 6.2 Ki 2
PGMNDAZLZGOWHP 6.2 Ki 5
PLVZHOWVQHWPON 6.2 IC50 4
YLSBAGZHIBFNRL 6.2 IC50 4
ZPEIMTDSQAKGNT 6.2 Ki 35 Yes
CUFJQHNVDRIQJL 6.2 Ki 5
FASDKYOPVNHBLU 6.2 Ki 5
GQGDLZJIYOGRNE 6.2 Ki 2
GYNZQBCSTGHPIZ 6.2 Ki 2
HTIRWRUKKGIFSB 6.2 Ki 2
IJELEDWFBGNAHO 6.2 Ki 2
IWCIBZDZIDMHMH 6.2 Ki 2
MFUWRMRKXKCSPL 6.2 Ki 2
SZOKTSDFOPVLFD 6.2 Ki 4 Yes
XYELHMUZUMBCJJ 6.2 Ki 2
YZDRSNBYBMAHDD 6.2 Ki 2
AIJIQCBYMBZLJD 6.2 Ki 6
IQDAWMWSGXPSNV 6.2 Ki 6
KAHXPONUPROIRS 6.2 Ki 7
QXYZJXCNTMMWEO 6.2 Ki 15
ZOAXAKJUBSMZJB 6.2 Ki 3
AKUFOSYLIYVIGY 6.1 Ki 2
CZLSEABFCZWLAR 6.1 Ki 4
FDMHBTAXJFCYLV 6.1 Ki 2
ISKSUBAAYHUDJC 6.1 Ki 4
YTSPXKNHGROQEX 6.1 Ki 4
ZSCRFGSBZVTGPQ 6.1 Ki 2
AELYPESLFOQFTR 6.1 Ki 4
BDECJFBHDUVJRU 6.1 Ki 6
CNXJBRGDAVLMOF 6.1 Ki 2
DATRLTNBZWRBPI 6.1 Ki 12
DMQUHZAYPOZSTL 6.1 Ki 2
FOCNVWPMXDBALZ 6.1 Ki 3
JSMDVVKGKQQXSH 6.1 Ki 4
KHUCESLAHQBKOQ 6.1 Ki 2
IPEQZSDWFQRQIF 6.1 Ki 2
2D structure