Target Details
UniProt ACP08908
Gene SymbolHTR1A
Protein Name5-hydroxytryptamine receptor 1A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 3,572
  • Clinical molecules 89
  • Avg pChEMBL 7.64
Top Co-occurrence Targets
Active Molecules (3,572)
InChIKey pChEMBL Type Targets Clinical
DGSJCQBCZUXHPR 9.1 Ki 4
AKXPLUFJRRUGNE 9.1 Ki 4
HCMVGFUNBPYWGU 9.1 Ki 3
PJBISDNIYJBREA 9.1 Ki 3
SLUWYSCSZRXUHY 9.1 Ki 3
BYJLEOXPONSXOY 9.1 Ki 5
LOKNTFKIZJDADX 9.1 Ki 3
ANCFDBAFLRCWEK 9.1 Ki 3
FUVSPPJJICMEMP 9.1 Ki 2
GSYXUBWRYIWXJK 9.1 Ki 2
IPGPPSLCUMESRR 9.1 Ki 4
PNRXQZLTVQCRMF 9.1 Ki 3
BZFUYHDDVGBTOS 9.1 Ki 2
DRHKJLXJIQTDTD 9.1 Ki 9
GOLUWUPEFVOPGA 9.1 IC50 3
GZRLRTFOHXYECM 9.1 Ki 4
HGEYJZMMUGWEOT 9.1 IC50 17
IUIOIGDUPSHYOT 9.1 IC50 2
IUVSEUFHPNITEQ 9.1 Ki 7
JRPAZCAZXFNBAT 9.1 Ki 4
MSFUUIPBIBJYNX 9.1 Ki 4
QCQQQZSWJWFIFV 9.1 Ki 4
RDTMBNGZUMUZNP 9.1 Ki 3
VPAUPKOMHDFAMG 9.1 Ki 4
VQMKNQCYRARFEO 9.1 Ki 3 Yes
WDBLAZNCHMHPRY 9.1 Ki 2
XKHJTHWUWGJDOX 9.1 Ki 9
YRAPNFDLJRSFKB 9.1 Ki 4
ZWIOIIOCCRESNK 9.1 Ki 4
ZYBLSQVXWVJACW 9.1 Ki 3
CNFSPPDVZAYHDT 9.1 Ki 4
JZMJEIJWBRTMLR 9.1 Ki 2
ULPHERUXCWNZNF 9.1 Ki 2
FIVZLAMKROFZLS 9.1 Ki 3
FZKSKVNYSCHGOF 9.1 Ki 2
IWHKEAOARZJLDH 9.1 Ki 2
STBHTUOPFMOXDX 9.1 Ki 3
XTIPDLJJVIOGHI 9.1 Ki 3
XZLUQCNWEIDMSJ 9.1 Ki 2
YZLCDNYSBSWVBY 9.1 Ki 4
ZKNQRQDTAWUUJL 9.1 Ki 4
ASFLUVKXUIJMQA 9.1 Ki 4
DFNUNBHMMOZMON 9.1 Ki 4
FFGYZWWOVBUEIV 9.1 Ki 3
KDBNOLRCLHHEBP 9.1 Ki 2 Yes
NUHXXOFRYNFFKK 9.1 Ki 4
AVSPJTOPUUMEGQ 9.1 Ki 3
CLADBLWFXVASRD 9.1 Ki 4
HPYBDVNCBKPJOQ 9.1 Ki 2
HSOIWCPMXCWYHB 9.1 Ki 2
2D structure