Target Details
UniProt ACP08908
Gene SymbolHTR1A
Protein Name5-hydroxytryptamine receptor 1A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 3,572
  • Clinical molecules 89
  • Avg pChEMBL 7.64
Top Co-occurrence Targets
Active Molecules (3,572)
InChIKey pChEMBL Type Targets Clinical
WBUCFEOIQMRVHB 9.4 Ki 9
WCPCVFLVWUACMN 9.4 Ki 2
WDDZPZKGLZNGEH 9.4 Ki 2
WNZKLSJSPOZSAM 9.4 Ki 4
WOMMHANJCVMKAZ 9.4 Ki 3
ZCYQPTKLMLTYQD 9.4 Ki 4
ZGKITGMYHCRUFD 9.4 Ki 7
BKRGVLQUQGGVSM 9.4 Ki 18
NBMCMVKIOBKUGI 9.4 Ki 3
PGGCRGAETLNAJC 9.4 Ki 11
GSTSDXKNOKALFJ 9.4 Ki 2
KYIGOCCCBXRHNJ 9.4 IC50 43
DSJDREDLRIFSQA 9.4 Ki 4
RRTCFJGKAMKAIY 9.4 Ki 14
SIINLBKMJGQYNO 9.4 Ki 3
BKRGVLQUQGGVSM 9.3 Ki 26 Yes
DUKNIHFTDAXJON 9.3 Ki 12
SMLCPNKOWBEDFF 9.3 Ki 3
GPDIVIMXUJNGLC 9.3 Ki 3
PYKXSNLYPSZMTQ 9.3 Ki 4
SGTFFUDLSDUTKM 9.3 Ki 4
GDZBFHVIKHSMAN 9.3 Ki 3
BILQJDKHRSUCQZ 9.3 Ki 5
BJVNWTOKTUJQCC 9.3 Ki 3
FMCRANLYZLAXGN 9.3 Ki 5
GCTKTFKNHOBZCQ 9.3 Ki 2
HFPMFXUJDFZECD 9.3 Ki 4
JGCUFOXBUYJGBX 9.3 Ki 3
NXQBRORDMXGPPG 9.3 Ki 2
OWOQRXHVMOMTJK 9.3 Ki 4
POZFPYZCVYTCQZ 9.3 Ki 2
QIJPXEALWJLAOE 9.3 Ki 9
SBDOPCIVOPZGMV 9.3 Ki 6
SIMNKURLSFAWDZ 9.3 Ki 8
SPYRKRZLYSXVFE 9.3 Ki 4
XJPPJJAODBUHAJ 9.3 Ki 4 Yes
ZBWVSTNZRBXPIP 9.3 Ki 4
HFWNGFIHHPNYEM 9.3 Ki 2
QHUHMRAZOMFJRX 9.3 Ki 4
JQTBIDKOADOXPE 9.3 Ki 2
LCZMXKRXXCYHBB 9.3 Ki 5
IRZUEVZANGAMPR 9.3 Ki 2 Yes
PJPXYNKEROPCAD 9.3 Ki 8
WOTQTCOGYGHNIU 9.3 Ki 3
MFUWMPKHVOQTMZ 9.3 Ki 2
GZRLRTFOHXYECM 9.2 Ki 4
VFNSXXVAZKMPQN 9.2 Ki 4
SCTHKCGXMXTKHG 9.2 Ki 4
UTVCJNNRVXMBSF 9.2 Ki 3
ZCYQPTKLMLTYQD 9.2 Ki 4
2D structure