Target Details
UniProt ACP08908
Gene SymbolHTR1A
Protein Name5-hydroxytryptamine receptor 1A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 3,572
  • Clinical molecules 89
  • Avg pChEMBL 7.64
Top Co-occurrence Targets
Active Molecules (3,572)
InChIKey pChEMBL Type Targets Clinical
BXPJDTCYZQOTIA 11.0 Ki 3
RVISYUPDXKKJLS 10.8 Ki 3
OLBJQOJHPPLFHK 10.5 Ki 2
BZPQHANIFQTYHQ 10.5 Ki 3
YOAVLBDWCVGCKZ 10.5 Ki 3
UHNTXNSIJZQVSR 10.3 Ki 3
QKQGOJLWKYGOGZ 10.3 Ki 3
VGNJZLFABGNCBA 10.3 Ki 2
DXWRIDGYFFSIIY 10.2 Ki 2
FRMZDOIYBVOLRB 10.2 Ki 7
ZMEGJWWPDKBOER 10.2 Ki 2
FFCUBEJNESQWBX 10.1 Ki 4
FOQOXYFYHFUCMT 10.1 Ki 3
FOQOXYFYHFUCMT 10.1 Ki 3
GPCOZCFGTRWRLE 10.1 Ki 3
GWAMGWDJCYIREE 10.1 Kd 20
IWBMAAUPHUCYCI 10.1 Kd 20
JAELRPUWEUXJPW 10.1 Ki 5
JZCAGBINSPHSNG 10.1 Ki 2
LMIGPJJYYRXPJA 10.1 Ki 4
MODBIBJHAWXYOZ 10.1 Kd 20
UKAZUPHMMINRDF 10.1 Ki 3
ZRQMUCDHVVOENY 10.1 Kd 17
LBGPXUXLKXFCMK 10.1 Ki 2
ZWIZEAIJEJNAJL 10.1 Ki 2
HCCHXMMABQRBMV 10.0 Ki 3
GQUKVOGAZWDTMK 10.0 Ki 2
GTEYGWXMYSXCRZ 10.0 Ki 5
IKMGSOGDZPNUTQ 10.0 Ki 3
KOWBAFDEMIDBCY 10.0 Ki 2
KXHGSYJSIPFIRS 10.0 Ki 4
MFXLHBQIIUCFFZ 10.0 Ki 2
SKSOBHHSERUEOI 10.0 IC50 3
SXCVVYUSUGUSMW 10.0 Ki 14
WDDZPZKGLZNGEH 10.0 Ki 2
JVMBIOQCKALKPB 10.0 Ki 4
FEPNYAFFRMEINW 10.0 Ki 3
TVCLMCWUAJMAEI 9.9 Ki 4
FFZUWXZVFRDGLT 9.9 Ki 3
ZKIAIYBUSXZPLP 9.9 Ki 29
BSRXZCMRRHEYBS 9.9 Ki 5
DHKSBFZUOUSCJC 9.9 Ki 4
DWJGZXZILMOEGQ 9.9 Ki 4
LHWYHPOPXMPQGV 9.9 Ki 4
RKTWFMDUKBINRA 9.9 Ki 5
XWFYCUBZTUUOJK 9.9 Ki 4
FGBDGNKVRNLYDB 9.9 Ki 4
QCTMCGZINYAROF 9.9 Ki 4
SPJPXOJVCGSOOK 9.9 IC50 5
JAAHNPXYHPFVSN 9.8 Ki 3
2D structure