Target Details
| UniProt AC | P08648 |
|---|---|
| Gene Symbol | ITGA5 |
| Protein Name | Integrin alpha-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (21)
- Arrhythmogenic right ventricular cardiomyopathy
- Bacterial invasion of epithelial cells
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pertussis
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Shigellosis
- Virion - Herpesvirus
- Yersinia infection
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VRTNUMBPIBDYLD
|
6.1 | IC50 | 5 | — | |
CVFCIUNYJXEWIG
|
6.1 | IC50 | 5 | — | |
HGFOOLONGOBCMP
|
6.1 | IC50 | 6 | — | |
LSAHZFHCOBEICB
|
6.1 | IC50 | 4 | — | |
ACHJOQIILIANHB
|
6.1 | IC50 | 4 | — | |
BWTVNRVTJZZPIR
|
6.1 | IC50 | 4 | — | |
WYTVCQXHVKVZEJ
|
6.1 | IC50 | 4 | — | |
ZJLLVRHQFNOZTN
|
6.1 | IC50 | 3 | — | |
BYQHRPBGTMGOIJ
|
6.0 | IC50 | 2 | — | |
VTZMVMKHYIBVPC
|
6.0 | IC50 | 3 | — | |
VXWPHQRTNDOPIH
|
6.0 | IC50 | 2 | — | |
UNRGZLRGJNKHCM
|
6.0 | IC50 | 5 | — | |
JUVWMVYEUFVLOP
|
6.0 | IC50 | 4 | — | |
XGLXZTFJSOLCED
|
6.0 | IC50 | 2 | — | |
YINCHOOHNDSILR
|
6.0 | IC50 | 4 | — | |
BLLLAUHTNAVSQR
|
6.0 | IC50 | 5 | — |