Target Details
| UniProt AC | P08648 |
|---|---|
| Gene Symbol | ITGA5 |
| Protein Name | Integrin alpha-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (21)
- Arrhythmogenic right ventricular cardiomyopathy
- Bacterial invasion of epithelial cells
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pertussis
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Shigellosis
- Virion - Herpesvirus
- Yersinia infection
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IOQRWBKYEFBRMN
|
6.3 | IC50 | 2 | — | |
KRRAGDWAJLZINA
|
6.3 | IC50 | 2 | — | |
LFBYRHNJGDKWKR
|
6.3 | IC50 | 2 | — | |
LWNVRRLYEWEYCH
|
6.3 | IC50 | 2 | — | |
LWPORHPDJGXVMO
|
6.3 | IC50 | 2 | — | |
NBFYQDLZBZGXPB
|
6.3 | IC50 | 4 | — | |
PAXYMJSURQLQAW
|
6.3 | IC50 | 2 | — | |
RLVWHKYTSBZABY
|
6.3 | IC50 | 3 | — | |
SXKPBPZVSACQSN
|
6.3 | IC50 | 3 | — | |
TUXAORRGUIOJAM
|
6.3 | IC50 | 2 | — | |
TXDUNPFVQQSUTP
|
6.3 | IC50 | 3 | — | |
UHXBOYLWYUPYDA
|
6.3 | IC50 | 3 | — | |
UXCIVWRENWMDLO
|
6.3 | IC50 | 2 | — | |
VMXDSWMLXPSSCM
|
6.3 | IC50 | 3 | — | |
VTJZZOUBHILYBS
|
6.3 | IC50 | 4 | — | |
WWAGHGZWLQKHTA
|
6.3 | IC50 | 2 | — | |
XFHCUQCLLGVBIK
|
6.3 | IC50 | 3 | — | |
XUZYXUYMPMIJCS
|
6.3 | IC50 | 2 | — | |
ZEDVVTNZWFMRKR
|
6.3 | IC50 | 3 | — | |
ZYXVFEGWGYFGOG
|
6.3 | IC50 | 2 | — | |
JBCUWZUACLSOTF
|
6.3 | IC50 | 2 | — | |
IGRZOKIVRZOBLQ
|
6.3 | IC50 | 4 | — | |
OAAQLWCJRCWASU
|
6.3 | IC50 | 2 | — | |
VOHFXKNBMJXQTC
|
6.3 | IC50 | 2 | — | |
XNQBUAXVSJPQJY
|
6.3 | IC50 | 2 | — | |
YBADCZRQGLGRGX
|
6.3 | IC50 | 2 | — | |
JQJLVAXZJTYVQY
|
6.2 | IC50 | 4 | — | |
ZONWPEAFLDQJPL
|
6.2 | IC50 | 6 | — | |
FVIAXINNEOEZCZ
|
6.2 | IC50 | 6 | — | |
LORYPHNOOIUAQG
|
6.2 | IC50 | 2 | — | |
WAJIHESGSSDZLV
|
6.2 | IC50 | 6 | — | |
AVAGDMNSAIAKBL
|
6.2 | IC50 | 3 | — | |
CPLSKPXBSSVARR
|
6.2 | IC50 | 3 | — | |
DRNAKEUEIWVLBV
|
6.2 | IC50 | 3 | — | |
GLAPOVNKDGONRS
|
6.2 | IC50 | 4 | — | |
IYDOQPMEINDDIU
|
6.2 | IC50 | 4 | — | |
PCZKSCFYEHCLNY
|
6.2 | IC50 | 3 | — | |
PNKBWMFDXVFJCQ
|
6.2 | IC50 | 3 | — | |
RSXKUDHUICLXQJ
|
6.2 | IC50 | 3 | — | |
UIUXPBJXTNSKSS
|
6.2 | IC50 | 3 | — | |
VNECHKYIECIXLL
|
6.2 | IC50 | 3 | — | |
WFUKISJPCINNHD
|
6.2 | IC50 | 3 | — | |
XDXCCFXTQYSODJ
|
6.2 | IC50 | 3 | — | |
ZHVJYOAURCOISG
|
6.2 | IC50 | 3 | — | |
WEXQBLSMARBRMG
|
6.2 | IC50 | 6 | — | |
ICTXJDJNDUREMP
|
6.2 | IC50 | 3 | — | |
JQEZMOGAXNWFSH
|
6.2 | IC50 | 2 | — | |
YLVNILLAZOYHHS
|
6.2 | IC50 | 6 | — | |
ZSEXNBSYJGXEIW
|
6.1 | IC50 | 7 | — | |
UKHTYQDNRXRVQA
|
6.1 | IC50 | 3 | — |