Target Details
| UniProt AC | P08648 |
|---|---|
| Gene Symbol | ITGA5 |
| Protein Name | Integrin alpha-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (21)
- Arrhythmogenic right ventricular cardiomyopathy
- Bacterial invasion of epithelial cells
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pertussis
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Shigellosis
- Virion - Herpesvirus
- Yersinia infection
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GRHCYZBYNORHKC
|
6.8 | IC50 | 4 | — | |
KDVWFGZFEJOVIX
|
6.8 | IC50 | 4 | — | |
MDCSKKRHLAAXNA
|
6.8 | IC50 | 2 | — | |
MKXYXLLDTVYISF
|
6.8 | IC50 | 2 | — | |
VFVGVPLUVIXFKU
|
6.8 | IC50 | 4 | — | |
NNGZKLHXGWZBQW
|
6.8 | IC50 | 4 | — | |
OQDKBZBKHWYBSI
|
6.8 | IC50 | 3 | — | |
RAFNWGJYLZVXFV
|
6.8 | IC50 | 5 | — | |
XOZRHQVPPRGARQ
|
6.8 | IC50 | 2 | — | |
BSJOIRBVGVDOJC
|
6.8 | IC50 | 3 | — | |
DVHYCJSDRSSPME
|
6.8 | IC50 | 4 | — | |
FXYDXLJEJBXFBD
|
6.7 | IC50 | 7 | — | |
HKOMVWLUPCUKGC
|
6.7 | IC50 | 2 | — | |
LDVWGBGQDNJFFY
|
6.7 | IC50 | 4 | — | |
RTSICEKVZOJTRJ
|
6.7 | IC50 | 2 | — | |
ZJQXQBNPHQGXKR
|
6.7 | IC50 | 2 | — | |
QIUVOSJLYMTVAE
|
6.7 | IC50 | 5 | — | |
FRXCQHJSACJLPG
|
6.7 | IC50 | 4 | — | |
NBIFCEAIUJPYTM
|
6.7 | IC50 | 2 | — | |
PRUCOWVKLZWPSA
|
6.7 | IC50 | 3 | — | |
BNEDPHPIEQKOBX
|
6.6 | IC50 | 4 | — | |
FFZRIJWHHIJYHI
|
6.6 | IC50 | 4 | — | |
YMYRFEUQHZOVAB
|
6.6 | IC50 | 2 | — | |
FMXCDFVBSWABHQ
|
6.6 | IC50 | 3 | — | |
DONYTUFIXISVKJ
|
6.6 | IC50 | 2 | — | |
QHCIXBBIFMPYIS
|
6.5 | IC50 | 2 | — | |
MANPFXQOUPQAJD
|
6.5 | IC50 | 3 | — | |
FEBHCRJBENHQJT
|
6.5 | IC50 | 4 | — | |
JVAQDGLFINTCRG
|
6.5 | IC50 | 2 | — | |
ZMKZFZRVGGPCLB
|
6.4 | IC50 | 2 | — | |
HMOIMLFTJZBAGO
|
6.4 | IC50 | 3 | — | |
BWOKYFQNZCEABS
|
6.4 | IC50 | 3 | — | |
PQWRZQIWMNBRRU
|
6.4 | IC50 | 3 | — | |
DZZGXQVCGKJMNH
|
6.4 | IC50 | 4 | — | |
HIKCELHIZSKMGI
|
6.4 | IC50 | 5 | — | |
QQGUOHQFMOOCJJ
|
6.4 | IC50 | 2 | — | |
XTNLRPMBRFOVIZ
|
6.4 | IC50 | 2 | — | |
NYBIVSZISCEEHW
|
6.4 | IC50 | 4 | — | |
SIVAZRUSFYJFGM
|
6.4 | IC50 | 3 | — | |
ZBCMRNQAMJVHOG
|
6.4 | IC50 | 4 | — | |
CNPLKUGUUWSZIK
|
6.3 | IC50 | 2 | — | |
DLORZJRWPLTLNY
|
6.3 | IC50 | 2 | — | |
AKXRNGZFXODFCT
|
6.3 | IC50 | 6 | — | |
DBNZZRMTJNJPLM
|
6.3 | IC50 | 2 | — | |
SXIKNOJEFQXCPA
|
6.3 | IC50 | 4 | — | |
KRNPACMXJWBKFZ
|
6.3 | IC50 | 2 | — | |
AJZHUKFTTKIGAR
|
6.3 | IC50 | 3 | — | |
BHDQCURWNGKMND
|
6.3 | IC50 | 2 | — | |
BIWLMYQUTFMBFS
|
6.3 | IC50 | 3 | — | |
CKPFLCVDCRYWAY
|
6.3 | IC50 | 3 | — |