Target Details
| UniProt AC | P08648 |
|---|---|
| Gene Symbol | ITGA5 |
| Protein Name | Integrin alpha-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (21)
- Arrhythmogenic right ventricular cardiomyopathy
- Bacterial invasion of epithelial cells
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pertussis
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Shigellosis
- Virion - Herpesvirus
- Yersinia infection
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LMCAPKVVZZHYLE
|
7.0 | IC50 | 5 | — | |
XIHSFCHJUDBZKE
|
7.0 | IC50 | 3 | — | |
KXLRYMPSHOVNJE
|
7.0 | IC50 | 6 | — | |
QEWKBLVMROGVIO
|
7.0 | IC50 | 6 | — | |
XGMBDTKPGSGTQW
|
7.0 | IC50 | 4 | — | |
BPTWIXQUGNKCHT
|
7.0 | IC50 | 4 | — | |
AICBXHQRXOXRSL
|
7.0 | IC50 | 4 | — | |
VDXWNRXEYNGPST
|
7.0 | IC50 | 4 | — | |
NEEFZJDFXACOOY
|
7.0 | IC50 | 4 | — | |
QQLUALUDFDCTAP
|
7.0 | IC50 | 2 | — | |
WXSLOTVKKDWKQR
|
7.0 | IC50 | 4 | — | |
YFKSRHSJFVAXDN
|
7.0 | IC50 | 2 | — | |
RSPFMOVFUKBJRO
|
7.0 | IC50 | 2 | — | |
FAEHBENUBLUAIB
|
6.9 | IC50 | 2 | — | |
GQBLOQLGKPVDDP
|
6.9 | IC50 | 2 | — | |
YBGMAGXRECTCHQ
|
6.9 | IC50 | 4 | — | |
ACAKBZZHDIANCL
|
6.9 | IC50 | 4 | — | |
PSZYZEZKPQGGPA
|
6.9 | IC50 | 6 | — | |
SXOHFYRRZAGKRM
|
6.9 | IC50 | 4 | — | |
KIOBNTPONYOMJE
|
6.9 | IC50 | 4 | — | |
MFVBSMYEXLRRIU
|
6.9 | IC50 | 5 | — | |
NVHPXYIRNJFKTE
|
6.9 | IC50 | 6 | — | |
UEDXMRKTOKTYSH
|
6.9 | IC50 | 3 | — | |
RRPRWSUXQMFYCJ
|
6.9 | IC50 | 3 | — | |
BSLQJJPIELRITP
|
6.8 | IC50 | 7 | — | |
FKASXWSDVMDKSE
|
6.8 | IC50 | 2 | — | |
LBMGZTODNZDURL
|
6.8 | IC50 | 2 | — | |
FRLFLFWXQJDPEU
|
6.8 | IC50 | 3 | — | |
GVGUPQRRZKSMPE
|
6.8 | IC50 | 3 | — | |
IDLRLZKYIBXZJD
|
6.8 | IC50 | 4 | — | |
ISTYMXNQOZXIPN
|
6.8 | IC50 | 3 | — | |
ITUSCLRGOZYBSW
|
6.8 | IC50 | 3 | — | |
JXMJWKSIBSTJIF
|
6.8 | IC50 | 3 | — | |
LGXRBPOHXLBIKM
|
6.8 | IC50 | 3 | — | |
MLVJCTIWVYAXRI
|
6.8 | IC50 | 3 | — | |
NYIJVOPSVVFNKF
|
6.8 | IC50 | 3 | — | |
OEPVDEQVNNISKB
|
6.8 | IC50 | 4 | — | |
OLYGJMIIGKIKIG
|
6.8 | IC50 | 3 | — | |
PVUNJFDGIRQSRE
|
6.8 | IC50 | 3 | — | |
QELQEUKCMHKXAF
|
6.8 | IC50 | 3 | — | |
QLQWVDXKTCOBFF
|
6.8 | IC50 | 3 | — | |
SXHBIHNIKMXDBA
|
6.8 | IC50 | 3 | — | |
UYMOSJMAWDJBMJ
|
6.8 | IC50 | 3 | — | |
VVRXUTAYELKZGA
|
6.8 | IC50 | 3 | — | |
VWJRHICPKCXJIR
|
6.8 | IC50 | 3 | — | |
WRAPGMNNYFJAFF
|
6.8 | IC50 | 3 | — | |
XTNCVSRPUAXOII
|
6.8 | IC50 | 2 | — | |
YELAOQDTELRPSE
|
6.8 | IC50 | 3 | — | |
YJLXHQJWGPXYIB
|
6.8 | IC50 | 5 | — | |
ZSMGYPDQBQVUFI
|
6.8 | IC50 | 3 | — |