Target Details
| UniProt AC | P08648 |
|---|---|
| Gene Symbol | ITGA5 |
| Protein Name | Integrin alpha-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (21)
- Arrhythmogenic right ventricular cardiomyopathy
- Bacterial invasion of epithelial cells
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pertussis
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Shigellosis
- Virion - Herpesvirus
- Yersinia infection
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GASMFAZDFTXBTB
|
7.4 | IC50 | 4 | — | |
KCNHHQRQBVCSLO
|
7.4 | IC50 | 4 | — | |
PXLVREINRJDXEF
|
7.4 | IC50 | 4 | — | |
XOCIVSKNARLKGI
|
7.4 | IC50 | 4 | — | |
AYRVAWFOHYBCGQ
|
7.4 | IC50 | 4 | — | |
BMHOPYDAWFKHEW
|
7.4 | IC50 | 3 | — | |
MIFZAPHWMCAHQZ
|
7.4 | IC50 | 5 | — | |
LPWSHOGTPIIOBC
|
7.4 | IC50 | 5 | — | |
WYPGVVZBOCXSCK
|
7.4 | IC50 | 4 | — | |
LFJKKQPLVRUFPC
|
7.4 | IC50 | 4 | — | |
PWDSDBVBKCIRHN
|
7.4 | IC50 | 4 | — | |
QYKHSZCOMAXNCJ
|
7.3 | IC50 | 6 | — | |
FAUUZARDASUJGS
|
7.3 | IC50 | 2 | — | |
RQGAXIDPYFPPMW
|
7.3 | IC50 | 4 | — | |
XFNZYXKVDFJAFI
|
7.3 | IC50 | 6 | — | |
RIRSYRXZEYNCLO
|
7.3 | IC50 | 4 | — | |
PDJSBAOCILQASK
|
7.3 | IC50 | 3 | — | |
RSPIDHXLVXDISW
|
7.3 | IC50 | 2 | — | |
HZLFZIQTWBACFC
|
7.3 | IC50 | 2 | — | |
WORXKOOYMZPIGP
|
7.3 | IC50 | 4 | — | |
CCFUBKFBAQEAGV
|
7.2 | IC50 | 4 | — | |
CCFUBKFBAQEAGV
|
7.2 | IC50 | 4 | — | |
CCFUBKFBAQEAGV
|
7.2 | IC50 | 2 | — | |
FDEYYGVHDVBTNW
|
7.2 | IC50 | 4 | — | |
JUCATPBOBDBSCE
|
7.2 | IC50 | 4 | — | |
DLJDTWYGOQOTKA
|
7.2 | IC50 | 3 | — | |
KXYAXQVLPNBUFO
|
7.2 | IC50 | 5 | — | |
JAUWZXFLIUKTGH
|
7.2 | Ki | 4 | — | |
PGMTXWDCGBRTJD
|
7.2 | IC50 | 2 | — | |
YJVQTPGCEVENKR
|
7.2 | IC50 | 4 | — | |
FUBVRQRCBDJFQQ
|
7.2 | IC50 | 6 | — | |
MHKXMNCZAAKYLC
|
7.2 | IC50 | 2 | — | |
CDROWTZQLMBXDQ
|
7.2 | IC50 | 4 | — | |
NKIPTRIPXHQDGW
|
7.2 | IC50 | 6 | — | |
FLTIMXZSLYRKOV
|
7.1 | IC50 | 6 | — | |
UXIFXRPPOKZVPG
|
7.1 | IC50 | 2 | — | |
SXIKNOJEFQXCPA
|
7.1 | IC50 | 4 | — | |
XXVHVXVVXGOJQZ
|
7.1 | IC50 | 4 | — | |
CVAFKDVZZYLXCZ
|
7.1 | IC50 | 6 | — | |
HOXLTGNIFJUOIA
|
7.1 | IC50 | 6 | — | |
XBZCXNWBZFZRPR
|
7.1 | IC50 | 2 | — | |
AYXKDCNGRBXXLP
|
7.1 | IC50 | 4 | — | |
BDFHRUNNBXEXIG
|
7.1 | IC50 | 2 | — | |
PQPGXHCKTBRKTN
|
7.1 | IC50 | 4 | — | |
QYOKHKZTOCBBQY
|
7.1 | IC50 | 5 | — | |
ROFCWWUBJHHVGZ
|
7.1 | IC50 | 6 | — | |
ZRRDVEJNFGIFLZ
|
7.1 | IC50 | 4 | — | |
TWZMXULIICKEJC
|
7.0 | IC50 | 4 | — | |
LGMXGJOVGIKKKC
|
7.0 | IC50 | 4 | — | |
SZBGXIGBOYKYGD
|
7.0 | IC50 | 2 | — |