Target Details
| UniProt AC | P08648 |
|---|---|
| Gene Symbol | ITGA5 |
| Protein Name | Integrin alpha-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (21)
- Arrhythmogenic right ventricular cardiomyopathy
- Bacterial invasion of epithelial cells
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pertussis
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Shigellosis
- Virion - Herpesvirus
- Yersinia infection
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DKGATRXTJTUOON
|
7.8 | IC50 | 3 | — | |
XWMGBLCMRLASDS
|
7.8 | IC50 | 8 | — | |
BIEDRWCJOCDGPG
|
7.7 | IC50 | 4 | — | |
CRYKFAHXDBDCDF
|
7.7 | IC50 | 2 | — | |
PGTXPSMKFDYRPN
|
7.7 | IC50 | 2 | — | |
UQYFVSMGEHOGBU
|
7.7 | IC50 | 5 | — | |
JNSJYLADRXNURW
|
7.7 | IC50 | 2 | — | |
LHCLWEHLDOMAOL
|
7.7 | IC50 | 2 | — | |
ZPLWVCHCWZALGS
|
7.7 | IC50 | 4 | — | |
LNRANMOOBUMBQZ
|
7.7 | IC50 | 2 | — | |
HAWHNGUKUZPYEE
|
7.7 | IC50 | 4 | — | |
QYKHSZCOMAXNCJ
|
7.7 | IC50 | 5 | — | |
RKBFMHGYXWQNKU
|
7.7 | IC50 | 4 | — | |
HKLGBIAIHDSNGD
|
7.7 | IC50 | 3 | — | |
UWPKDZSNCCHXJT
|
7.7 | IC50 | 4 | — | |
CJYMQDSGVRJJGX
|
7.7 | IC50 | 4 | — | |
HOJQNBKLKYCOIL
|
7.7 | IC50 | 6 | — | |
QKCFDPUKGKJIML
|
7.7 | IC50 | 7 | — | |
RZYRWEAZPQSSKX
|
7.7 | IC50 | 5 | — | |
ZJLJEWROVSZOMN
|
7.7 | IC50 | 6 | — | |
CFUKCNIRQBDDDD
|
7.6 | IC50 | 2 | — | |
FEOYKJVLQOYKSD
|
7.6 | IC50 | 4 | — | |
ILLZNYBFYMXUGH
|
7.6 | IC50 | 2 | — | |
JBCUWZUACLSOTF
|
7.6 | IC50 | 4 | — | |
QKJVOACJWLIFLA
|
7.6 | IC50 | 4 | — | |
DEASIAFXABQVBE
|
7.6 | IC50 | 2 | — | |
DGXVRVIKQDYUDK
|
7.6 | IC50 | 3 | — | |
HNKFTNWKBPAXKF
|
7.6 | IC50 | 4 | — | |
UMZVBZDHGKJFGQ
|
7.6 | IC50 | 5 | — | |
IPLLAQOFEDGGKD
|
7.6 | IC50 | 4 | — | |
PVQYTVXYFKKNTQ
|
7.6 | IC50 | 4 | — | |
UQEWVVUNGPKKKR
|
7.6 | IC50 | 6 | — | |
XXBNSEBYSGKBAQ
|
7.6 | IC50 | 4 | — | |
VHOAQASXQVEHKS
|
7.6 | IC50 | 2 | — | |
JYJNRUFKUMSRIN
|
7.5 | IC50 | 6 | — | |
QNWRGRATEXLYQY
|
7.5 | Ki | 2 | — | |
RURWNESJHWLUMA
|
7.5 | IC50 | 3 | — | |
NWOOORGYRVRDTD
|
7.5 | IC50 | 4 | — | |
UPRAJHBYWOGILD
|
7.5 | IC50 | 2 | — | |
YUFZLCHTKCDKMO
|
7.5 | IC50 | 4 | — | |
ZMKLPAJURKFWIQ
|
7.5 | IC50 | 5 | — | |
MGRPJUCLIBBWKX
|
7.5 | IC50 | 2 | — | |
QJPJMPQXWLLPPI
|
7.5 | IC50 | 4 | — | |
IVVOOUBTAXUXMJ
|
7.5 | IC50 | 2 | — | |
IFDCMTYFWOPBHL
|
7.5 | IC50 | 2 | — | |
KTPKPDHZXPMGRV
|
7.4 | IC50 | 5 | — | |
LOXDBHIFADBELN
|
7.4 | IC50 | 7 | — | |
MAQNBVXADCFFPW
|
7.4 | IC50 | 4 | — | |
ZDSIXCUNSXFSMQ
|
7.4 | IC50 | 6 | — | |
AGSQFOYLHPCNBU
|
7.4 | IC50 | 2 | — |