Target Details
| UniProt AC | P08648 |
|---|---|
| Gene Symbol | ITGA5 |
| Protein Name | Integrin alpha-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (21)
- Arrhythmogenic right ventricular cardiomyopathy
- Bacterial invasion of epithelial cells
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pertussis
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Shigellosis
- Virion - Herpesvirus
- Yersinia infection
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OURYZIAAXSSBIO
|
8.4 | IC50 | 5 | — | |
CJFKBQRLRONQOT
|
8.3 | IC50 | 7 | — | |
RBJQMIIPTLTYFP
|
8.3 | IC50 | 8 | — | |
ZMXBIIQMSGOIRZ
|
8.3 | Kd | 7 | — | |
IWUIDYZQPXSVJK
|
8.3 | IC50 | 2 | — | |
UXIFXRPPOKZVPG
|
8.3 | IC50 | 4 | — | |
WMAYUSHYHMSHFY
|
8.3 | IC50 | 6 | — | |
WMAYUSHYHMSHFY
|
8.3 | IC50 | 4 | — | |
ACYKBAYFNYDVSD
|
8.2 | IC50 | 2 | — | |
PJJWGMOYKFOUPO
|
8.2 | IC50 | 5 | — | |
RCCYAIQAQJPLAH
|
8.2 | IC50 | 3 | — | |
XRIHUZYLIIDSBZ
|
8.2 | IC50 | 5 | — | |
IHCPRNUOVTWPFZ
|
8.2 | IC50 | 2 | — | |
WXSLOTVKKDWKQR
|
8.2 | IC50 | 2 | — | |
YBGMAGXRECTCHQ
|
8.1 | IC50 | 2 | — | |
CXHCNOMGODVIKB
|
8.1 | IC50 | 7 | — | |
ILKRHUYCJMCBRQ
|
8.1 | IC50 | 8 | — | |
AGSQFOYLHPCNBU
|
8.1 | IC50 | 2 | — | |
LMCAPKVVZZHYLE
|
8.1 | IC50 | 4 | — | |
XIHSFCHJUDBZKE
|
8.1 | IC50 | 2 | — | |
OVSFRNHGVCEDQP
|
8.1 | IC50 | 2 | — | |
XUISHROIRBHOIM
|
8.1 | IC50 | 4 | — | |
BSNWAPOUYOPCPS
|
8.0 | IC50 | 6 | — | |
DPXBPHOGQDXQKU
|
8.0 | IC50 | 2 | — | |
DQNUIKGZODIUGL
|
8.0 | IC50 | 2 | — | |
FFLMJKGHLKUKDV
|
8.0 | IC50 | 2 | — | |
IXFAGPXZKNFPLS
|
8.0 | IC50 | 2 | — | |
JESHEQMKKYQWKH
|
8.0 | IC50 | 4 | — | |
MHVNXFCJVCIDMA
|
8.0 | IC50 | 2 | — | |
MRGLCDMUTJGVNZ
|
8.0 | IC50 | 2 | — | |
PINWKOWMUAOTOO
|
8.0 | IC50 | 2 | — | |
RTHTZKFWJRGDKZ
|
8.0 | IC50 | 4 | — | |
SFCYQXKSWPPSIX
|
8.0 | IC50 | 4 | — | |
SNTLUFHEOMJBDE
|
8.0 | IC50 | 2 | — | |
VFNZJTWWZVYTGA
|
8.0 | IC50 | 4 | — | |
YINCHOOHNDSILR
|
8.0 | IC50 | 4 | — | |
SZBGXIGBOYKYGD
|
8.0 | IC50 | 2 | — | |
FUCDPKMSCYXLSE
|
8.0 | IC50 | 2 | — | |
HSSWSZWMLOODPR
|
7.9 | IC50 | 2 | — | |
HCCCRTKFBOCXHX
|
7.9 | IC50 | 2 | — | |
KVWSUPBEKULILJ
|
7.9 | IC50 | 4 | — | |
MDRYYKCWQBJPBJ
|
7.9 | IC50 | 3 | — | |
VVIGVXDFMPIPRO
|
7.9 | IC50 | 4 | — | |
YUBVJZGWIJZEGM
|
7.9 | IC50 | 5 | — | |
TZNXKIAIKROUOK
|
7.8 | IC50 | 4 | — | |
HKLGBIAIHDSNGD
|
7.8 | IC50 | 3 | — | |
LJKWPNDKPDWWIA
|
7.8 | IC50 | 4 | — | |
WKXPTLWKGRAHCK
|
7.8 | IC50 | 4 | — | |
YAXVKGQMOOKIMH
|
7.8 | IC50 | 4 | — | |
AMLYAMJWYAIXIA
|
7.8 | IC50 | 7 | — |