Target Details
| UniProt AC | P08648 |
|---|---|
| Gene Symbol | ITGA5 |
| Protein Name | Integrin alpha-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 366
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (21)
- Arrhythmogenic right ventricular cardiomyopathy
- Bacterial invasion of epithelial cells
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Herpes simplex virus 1 infection
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pertussis
- Phagosome
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Shigellosis
- Virion - Herpesvirus
- Yersinia infection
Active Molecules (366)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LRJXQAWFNQBGLZ
|
10.0 | IC50 | 5 | — | |
IBXMYCNAAVLIET
|
9.7 | IC50 | 4 | — | |
NIRVMUZGMXCWKU
|
9.7 | Ki | 2 | — | |
HXCIDANYYUBZDI
|
9.5 | IC50 | 2 | — | |
JXVVEFIKDDVLOS
|
9.5 | IC50 | 8 | — | |
KTSCJCLXFWHLBQ
|
9.4 | IC50 | 4 | — | |
YQOFOSAJQMWIAT
|
9.4 | IC50 | 4 | — | |
TXIWNLQFRATZFL
|
9.4 | Ki | 4 | — | |
GDEQKRGKHZOXGD
|
9.3 | IC50 | 8 | — | |
OBOJFQICXTYCRY
|
9.3 | IC50 | 8 | — | |
LMTFGZLYPXNJRU
|
9.3 | IC50 | 2 | — | |
LTEAZKWKEALJQD
|
9.3 | IC50 | 4 | — | |
ZWFUXTUZVCZUMC
|
9.3 | IC50 | 2 | — | |
MFCABRSSOZYCRL
|
9.2 | IC50 | 8 | — | |
PEFBVOAICYLSAF
|
9.2 | IC50 | 8 | — | |
QTBFGJFGHGTDRF
|
9.2 | IC50 | 8 | — | |
SHRSEUHJTZQLRO
|
9.2 | IC50 | 8 | — | |
PCEMPIMHMWVATP
|
9.2 | IC50 | 5 | — | |
RTYLRDWEJUNBLU
|
9.2 | IC50 | 8 | — | |
UDGWKAUBGPXUNT
|
9.2 | IC50 | 2 | — | |
YPAMHQMVIMQKOR
|
9.2 | IC50 | 8 | — | |
CJRDXSVCUSRJDR
|
9.1 | IC50 | 8 | — | |
HIKDGFUZLZJZCB
|
9.1 | IC50 | 8 | — | |
IPSRDFZOWABPRU
|
9.1 | IC50 | 4 | — | |
MYSBVCKSODARFZ
|
9.1 | IC50 | 3 | — | |
XLANGJRVQABTFO
|
9.1 | IC50 | 5 | — | |
BQYBIJDRTDZCAJ
|
9.0 | IC50 | 8 | — | |
BWAUVRFZNDRMLY
|
9.0 | IC50 | 8 | — | |
GFTVRPWYQDITLC
|
9.0 | IC50 | 5 | — | |
QLBXWVBTUGYSGI
|
9.0 | IC50 | 8 | — | |
RBJYKFLLCXRSGC
|
9.0 | Ki | 2 | — | |
VCAOZNYTIATHLZ
|
9.0 | Ki | 2 | — | |
XRXSSPOFDFFALK
|
9.0 | IC50 | 8 | — | |
ZAMKDPACDNUZPJ
|
9.0 | IC50 | 8 | — | |
CGSLGBRMSMBNMX
|
9.0 | IC50 | 6 | — | |
OMXIQNJVPRHGNN
|
8.8 | IC50 | 4 | — | |
SAFQBUKUEAMDGO
|
8.8 | IC50 | 3 | — | |
SMNXQFKEUFRQPU
|
8.8 | IC50 | 2 | — | |
PTCMVGOQRMWOTP
|
8.8 | IC50 | 4 | — | |
GNNSUMADLWATJP
|
8.8 | IC50 | 5 | — | |
AZJYXUVHLYXCJY
|
8.8 | IC50 | 2 | — | |
AZJYXUVHLYXCJY
|
8.8 | IC50 | 2 | — | |
SQTQEWRATPPDHW
|
8.8 | IC50 | 3 | — | |
UEBUMZGZKUPTHB
|
8.8 | IC50 | 4 | — | |
UZVROHMMUDQAOJ
|
8.8 | IC50 | 5 | — | |
NAGIMKJAUDLRFH
|
8.7 | IC50 | 4 | — | |
UCBYYQWMMNUSGH
|
8.7 | IC50 | 8 | — | |
LKEWELOHCDVPMS
|
8.6 | IC50 | 4 | — | |
KJPQVMIRPSWAHV
|
8.5 | Ki | 2 | — | |
JIYOXFLRVUFAQT
|
8.5 | IC50 | 2 | — |