Target Details
| UniProt AC | P08631 |
|---|---|
| Gene Symbol | HCK |
| Protein Name | Tyrosine-protein kinase HCK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 379
- Clinical molecules 191
- Avg pChEMBL 7.22
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (379)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZXLCCABWVQDAOS
|
6.1 | IC50 | 3 | Yes | |
UORAPQCBWYIISR
|
6.1 | IC50 | 15 | — | |
DINPOPQNCDTVPQ
|
6.1 | IC50 | 10 | Yes | |
IZVDYFCDVQANSW
|
6.1 | IC50 | 3 | — | |
PTTXMHGPBHSAPT
|
6.1 | IC50 | 5 | Yes | |
DSBZQMQVJJPSIP
|
6.1 | IC50 | 2 | — | |
CMUZPNXYCOKJJJ
|
6.1 | IC50 | 7 | Yes | |
HKWNGVFHUCRTTQ
|
6.1 | IC50 | 7 | Yes | |
SAMCEVLBPWDZMX
|
6.1 | IC50 | 5 | Yes | |
ODPGGGTTYSGTGO
|
6.1 | Kd | 153 | — | |
QFUHCUNJMQVKME
|
6.1 | IC50 | 8 | Yes | |
WINHZLLDWRZWRT
|
6.1 | Kd | 201 | Yes | |
WXCKXLFOEBUZDO
|
6.1 | IC50 | 6 | Yes | |
FLBNLJLONKAPLR
|
6.0 | Kd | 31 | — | |
LNWUSIFVARIMOH
|
6.0 | IC50 | 6 | Yes | |
DAXMIVDYBBFSGN
|
6.0 | IC50 | 4 | — | |
GLYDCPPHXDVIKA
|
6.0 | IC50 | 5 | Yes | |
NHVGQRASKRTWLZ
|
6.0 | IC50 | 5 | Yes | |
ORVLOIUKTHUQPU
|
6.0 | IC50 | 5 | Yes | |
RCOGIBMVENMBNJ
|
6.0 | IC50 | 3 | — | |
AGEIBLLCZVGHLI
|
6.0 | IC50 | 9 | Yes | |
XLSPYLMTRXPYKY
|
6.0 | IC50 | 13 | — | |
ZZSBPGIGIUFJRA
|
6.0 | Kd | 46 | — | |
PYCBKUUFGVDPOF
|
6.0 | Ki | 4 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
LMVAHLFZGWUGNF
|
6.0 | IC50 | 8 | Yes | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
VMZGXVLGNHMKLW
|
6.0 | IC50 | 2 | Yes |