Target Details
| UniProt AC | P08631 |
|---|---|
| Gene Symbol | HCK |
| Protein Name | Tyrosine-protein kinase HCK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 379
- Clinical molecules 191
- Avg pChEMBL 7.22
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (379)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WLXHZMYOVDOALX
|
6.4 | IC50 | 5 | Yes | |
HGALDAPNHYJZAJ
|
6.4 | IC50 | 11 | Yes | |
PGXQNHGXDFCMOJ
|
6.4 | IC50 | 10 | Yes | |
FITNUKNIUJHPPH
|
6.4 | IC50 | 5 | Yes | |
FXCRGRHHHOSJRE
|
6.4 | IC50 | 5 | Yes | |
SHPFDGWALWEPGS
|
6.4 | Kd | 35 | — | |
WLLDKVYCGDHDLF
|
6.4 | IC50 | 6 | Yes | |
YFNWWNRZJGMDBR
|
6.4 | Kd | 35 | — | |
REZFVUNAFUHYBW
|
6.3 | IC50 | 5 | Yes | |
YCGAVAFYTUFYPA
|
6.3 | IC50 | 6 | Yes | |
NADBSABGTQOEQF
|
6.3 | IC50 | 2 | — | |
SRDCKXVGOFJLJK
|
6.3 | IC50 | 3 | Yes | |
IEIWIPIQYLVOCL
|
6.3 | IC50 | 3 | — | |
NITOVUIHLVISSN
|
6.3 | IC50 | 5 | Yes | |
SOLCZUBPADGMSF
|
6.3 | IC50 | 5 | Yes | |
JWNPDZNEKVCWMY
|
6.3 | Kd | 57 | Yes | |
FCNPQYHKUYSELK
|
6.3 | IC50 | 8 | — | |
SJKCAVNLLOXGJL
|
6.3 | Ki | 8 | — | |
CNWAVQYSQHXMCH
|
6.3 | IC50 | 3 | Yes | |
PJWDSDGNSMGWKJ
|
6.3 | IC50 | 4 | Yes | |
MLDQJTXFUGDVEO
|
6.3 | IC50 | 85 | Yes | |
AXQKJTHCYRYSLF
|
6.3 | IC50 | 3 | Yes | |
DBZCDBKTCUKQPQ
|
6.3 | IC50 | 8 | Yes | |
LTZAOEYIDIFFHJ
|
6.3 | IC50 | 5 | — | |
AMERZUAKIAGPBA
|
6.3 | IC50 | 7 | Yes | |
DPZGKYJHTOSMIA
|
6.3 | IC50 | 8 | — | |
GMQQMSKNSNVPOW
|
6.3 | IC50 | 9 | Yes | |
IBCGPVVKHZXWNX
|
6.3 | IC50 | 7 | — | |
KUCNBQPAJZRQMJ
|
6.3 | IC50 | 11 | — | |
KZRDVFBPXXGSPD
|
6.3 | IC50 | 9 | — | |
QUFURWJAQILIFO
|
6.3 | IC50 | 9 | — | |
KAANTKMOHHINMM
|
6.2 | IC50 | 4 | Yes | |
FLOXVEVSESQZRQ
|
6.2 | IC50 | 2 | Yes | |
XXJWYDDUDKYVKI
|
6.2 | Kd | 52 | — | |
IYVUNPAVFASLSV
|
6.2 | IC50 | 6 | Yes | |
PBCZSGKMGDDXIJ
|
6.2 | Kd | 68 | Yes | |
QPZURRPXZSPBJE
|
6.2 | IC50 | 9 | Yes | |
USVCWSAJUAARAL
|
6.2 | Kd | 8 | — | |
CTLVZTMBHKZFIR
|
6.2 | IC50 | 3 | — | |
HHFBDROWDBDFBR
|
6.2 | Ki | 40 | Yes | |
LOLPPWBBNUVNQZ
|
6.2 | Kd | 97 | Yes | |
LEODTNLMHLRQCI
|
6.2 | IC50 | 2 | — | |
BDGXAHBOBRAVIN
|
6.2 | IC50 | 3 | — | |
WJEOLQLKVOPQFV
|
6.2 | Kd | 24 | — | |
CSGQVNMSRKWUSH
|
6.2 | Kd | 21 | — | |
DHYADLCEAXMYPS
|
6.2 | IC50 | 9 | Yes | |
ICPHLXAHKNXIGM
|
6.2 | IC50 | 4 | Yes | |
BMGQWWVMWDBQGC
|
6.1 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.1 | Kd | 91 | Yes | |
DMXWTHVOLSODIU
|
6.1 | Ki | 4 | — |