Target Details
| UniProt AC | P08631 |
|---|---|
| Gene Symbol | HCK |
| Protein Name | Tyrosine-protein kinase HCK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 379
- Clinical molecules 191
- Avg pChEMBL 7.22
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (379)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MFAQYJIYDMLAIM
|
6.7 | Kd | 130 | Yes | |
NVHKWMBHTXQWRP
|
6.7 | IC50 | 9 | Yes | |
OBALKFHHXFROHH
|
6.7 | IC50 | 3 | — | |
RNRCLARSVNONBS
|
6.7 | IC50 | 3 | Yes | |
AILRADAXUVEEIR
|
6.7 | IC50 | 75 | — | |
DORRCVAXQFZOLU
|
6.7 | IC50 | 2 | — | |
JZTOUVBEZONDKA
|
6.7 | Ki | 80 | — | |
OSAWFUCUZJNEID
|
6.7 | IC50 | 20 | — | |
WINHZLLDWRZWRT
|
6.7 | Ki | 66 | — | |
IXWAAWQRRFJLQU
|
6.7 | IC50 | 3 | — | |
MXPLPMSWGMUSSK
|
6.7 | IC50 | 2 | — | |
MJOCJDMQRCJQJF
|
6.7 | IC50 | 7 | — | |
RUQMPILTACLXOK
|
6.7 | IC50 | 6 | Yes | |
DEFQAMZNXBZPPX
|
6.7 | IC50 | 2 | — | |
AYZBGELVIWCHIM
|
6.6 | IC50 | 5 | Yes | |
NVFPMSWRLJYMJE
|
6.6 | IC50 | 6 | — | |
QVFCDPRQRUAFKS
|
6.6 | IC50 | 10 | Yes | |
TXZDVQGUIJKUMP
|
6.6 | IC50 | 6 | Yes | |
NOVYSIQVVWXHGB
|
6.6 | IC50 | 3 | — | |
YOBIWCLAYQWPPW
|
6.6 | IC50 | 23 | — | |
FIENVLBRUWEWDS
|
6.6 | IC50 | 3 | Yes | |
XVTLRUAQTJKQLQ
|
6.6 | IC50 | 9 | Yes | |
NXSJMRCTGYTSTK
|
6.6 | Kd | 200 | — | |
UOKGZPYGRJDACN
|
6.6 | IC50 | 7 | Yes | |
YGTYIGUWQYTZMS
|
6.6 | IC50 | 5 | Yes | |
MDBPVHFMWKYINB
|
6.6 | IC50 | 3 | Yes | |
QRJVSLZNMWIKRS
|
6.6 | IC50 | 7 | Yes | |
UIARLYUEJFELEN
|
6.6 | Kd | 289 | Yes | |
MOSKATHMXWSZTQ
|
6.6 | IC50 | 16 | Yes | |
OSVUGUHRKMMBSE
|
6.5 | Kd | 170 | — | |
YRCHYHRCBXNYNU
|
6.5 | Kd | 13 | — | |
AAHKGRWRYBCWDL
|
6.5 | IC50 | 11 | Yes | |
PHVRYQBXECZHNT
|
6.5 | IC50 | 2 | — | |
BJNPYRHGWJVECX
|
6.5 | IC50 | 6 | Yes | |
CQZZCFVTEOJWAW
|
6.5 | IC50 | 5 | Yes | |
PDQSBODXIIIHSM
|
6.5 | IC50 | 3 | Yes | |
FVPBLAKABVRLRX
|
6.5 | IC50 | 9 | Yes | |
IBSCAHNKEHRFKF
|
6.5 | IC50 | 4 | Yes | |
JNIIGOXKPNCTTH
|
6.5 | IC50 | 4 | Yes | |
GMIVUSAKVGKIOC
|
6.5 | IC50 | 4 | Yes | |
YXLKDESGHOQYDJ
|
6.5 | IC50 | 3 | Yes | |
UHTHHESEBZOYNR
|
6.4 | Kd | 66 | Yes | |
YTSDNPLOCDVGNB
|
6.4 | IC50 | 8 | — | |
CXDDSIHNNLQHGV
|
6.4 | IC50 | 2 | — | |
DUPSNQFPAJUAKA
|
6.4 | IC50 | 9 | Yes | |
REDBMKRPRFVCHI
|
6.4 | IC50 | 4 | Yes | |
HHZIURLSWUIHRB
|
6.4 | Kd | 57 | Yes | |
JXJHMLMFXVHUJX
|
6.4 | IC50 | 2 | — | |
MCAASVHSHOYFNM
|
6.4 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
6.4 | Kd | 231 | Yes |