Target Details
| UniProt AC | P08631 |
|---|---|
| Gene Symbol | HCK |
| Protein Name | Tyrosine-protein kinase HCK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 379
- Clinical molecules 191
- Avg pChEMBL 7.22
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (379)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZTWYTYUOHYGWSG
|
7.1 | IC50 | 9 | Yes | |
DORRCVAXQFZOLU
|
7.1 | IC50 | 2 | — | |
HVUAYFFHDRNLOX
|
7.1 | IC50 | 11 | Yes | |
PNRBQMZDBPEICZ
|
7.1 | IC50 | 3 | — | |
JDFGIOCJMJJUNK
|
7.1 | IC50 | 6 | Yes | |
WVXNSAVVKYZVOE
|
7.1 | IC50 | 92 | — | |
FHNLPTRXVQOXQO
|
7.1 | IC50 | 7 | Yes | |
WSGHPGAVEJYWCS
|
7.1 | IC50 | 3 | Yes | |
GEZALMMCQYDFML
|
7.1 | IC50 | 15 | Yes | |
QPSCCNWGOLMGKW
|
7.1 | IC50 | 4 | Yes | |
WPXVVAWAHQHJPF
|
7.1 | IC50 | 41 | — | |
AULCRCVNIWNUTH
|
7.0 | IC50 | 10 | Yes | |
LCQAIZAFSOZWRC
|
7.0 | IC50 | 8 | Yes | |
BZYKWEQWEPHEQZ
|
7.0 | IC50 | 10 | Yes | |
OUKYUETWWIPKQR
|
7.0 | Kd | 31 | Yes | |
PTHVKCSYXICMAR
|
7.0 | IC50 | 14 | — | |
IAYGCINLNONXHY
|
7.0 | Kd | 50 | — | |
KUUPATHXUAIQFZ
|
7.0 | IC50 | 2 | — | |
ITENSOATZCMKDD
|
7.0 | IC50 | 3 | — | |
NXCRYXWTLYEUAS
|
7.0 | IC50 | 3 | Yes | |
XGALLCVXEZPNRQ
|
7.0 | IC50 | 39 | Yes | |
OUQOXXMJLDQZQC
|
7.0 | IC50 | 6 | Yes | |
BMPXPANSAQOTAY
|
6.9 | IC50 | 2 | — | |
DKZYXHCYPUVGAF
|
6.9 | Kd | 112 | — | |
QOYOSSAKTDDRJV
|
6.9 | IC50 | 11 | Yes | |
ULLIAFSPUSWCIL
|
6.9 | IC50 | 10 | Yes | |
DEFQAMZNXBZPPX
|
6.9 | IC50 | 2 | — | |
XJPZZAAKTVLITO
|
6.9 | IC50 | 3 | Yes | |
ITOYZJGFTNTKKR
|
6.9 | IC50 | 11 | Yes | |
VKGKEHUDLZDBMP
|
6.9 | IC50 | 5 | Yes | |
KUUPATHXUAIQFZ
|
6.9 | IC50 | 2 | — | |
UEJXELMBDCXXAQ
|
6.9 | IC50 | 9 | — | |
XKFTZKGMDDZMJI
|
6.9 | Kd | 64 | Yes | |
ZVIKAJOZJVAHPH
|
6.9 | IC50 | 5 | Yes | |
APPXQUDJLJXULP
|
6.8 | IC50 | 47 | — | |
WKDACQVEJIVHMZ
|
6.8 | Kd | 46 | — | |
LQIVXZFCXIBJSU
|
6.8 | IC50 | 10 | Yes | |
NHHQJBCNYHBUSI
|
6.8 | Kd | 220 | — | |
OYFMIXVMTCYDNY
|
6.8 | IC50 | 6 | Yes | |
SPUWUOGLPPVXCW
|
6.8 | IC50 | 15 | Yes | |
PIQCTGMSNWUMAF
|
6.8 | Ki | 137 | Yes | |
JXPFBRYPSJLQII
|
6.8 | IC50 | 3 | — | |
KLQFQJDEPBUNAK
|
6.8 | IC50 | 6 | Yes | |
FRBJLBMEOUWTOH
|
6.8 | IC50 | 3 | — | |
KOICAHGTHMWKIZ
|
6.8 | IC50 | 6 | Yes | |
YLLYKQYSOWECSZ
|
6.8 | IC50 | 4 | Yes | |
DAZCBQNFGSWSQG
|
6.7 | IC50 | 8 | Yes | |
GJAQIFQPFSPOOM
|
6.7 | IC50 | 2 | — | |
UBWALTPIDHCQBF
|
6.7 | IC50 | 3 | — | |
HHVUDVWMACNSOB
|
6.7 | IC50 | 4 | Yes |