Target Details
| UniProt AC | P08631 |
|---|---|
| Gene Symbol | HCK |
| Protein Name | Tyrosine-protein kinase HCK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 379
- Clinical molecules 191
- Avg pChEMBL 7.22
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (379)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GDQTYFYNHJDRBD
|
8.3 | IC50 | 2 | — | |
KTULYYQYBLJWBV
|
8.3 | IC50 | 2 | — | |
MRCFTWAYZAHAFA
|
8.3 | IC50 | 12 | Yes | |
MBPKPSDAPFPECJ
|
8.2 | IC50 | 12 | Yes | |
VEORWCZDRQSGJH
|
8.2 | IC50 | 10 | Yes | |
KSUDUUBCXJUFRL
|
8.2 | Kd | 12 | — | |
REFXTMLPVWSINW
|
8.2 | IC50 | 2 | — | |
ZCQBIMLCHPNRKB
|
8.2 | IC50 | 3 | — | |
POLFXOSYBGYACO
|
8.2 | IC50 | 2 | — | |
BMJIPGXVDYVSGD
|
8.2 | IC50 | 4 | — | |
IVZNWJUHDBLKKT
|
8.1 | IC50 | 2 | — | |
LNQHMSWBIGYWSY
|
8.1 | IC50 | 3 | — | |
XLRGWOQAKMIFSL
|
8.1 | IC50 | 2 | — | |
BMHCYYLFLWTPHZ
|
8.1 | IC50 | 4 | Yes | |
COAQRADEUYYCDG
|
8.1 | IC50 | 12 | Yes | |
DBXJNQABFNNKPN
|
8.1 | Kd | 7 | — | |
NVRXTLZYXZNATH
|
8.1 | IC50 | 47 | Yes | |
URQAXVPGUSETSW
|
8.1 | IC50 | 4 | — | |
COAQRADEUYYCDG
|
8.1 | IC50 | 12 | Yes | |
DPSNOZFUMXEANO
|
8.1 | Kd | 7 | — | |
CEUSZLVORFRBCV
|
8.1 | IC50 | 13 | — | |
HRRMXIICSWVXIS
|
8.1 | IC50 | 13 | Yes | |
KADWMAJVBHJWDX
|
8.1 | IC50 | 3 | — | |
KXTIIOOGQPWWGE
|
8.1 | IC50 | 6 | Yes | |
PFRDPPRTLFHGLR
|
8.1 | IC50 | 10 | Yes | |
CJMMCIXRPVLDBH
|
8.0 | IC50 | 12 | Yes | |
KMMUTXPSVYLUNZ
|
8.0 | IC50 | 3 | — | |
KTTGLAHMSDMRLJ
|
8.0 | IC50 | 12 | Yes | |
QYPSALIXKCRYNZ
|
8.0 | IC50 | 12 | Yes | |
RHFWTFDTRBFIHU
|
8.0 | IC50 | 13 | Yes | |
GIEDBGFYGHINFT
|
8.0 | IC50 | 8 | — | |
KUMLEJXITHSWSP
|
8.0 | IC50 | 9 | Yes | |
KUUPATHXUAIQFZ
|
8.0 | IC50 | 2 | — | |
PPCDZYRDXIKRDW
|
8.0 | IC50 | 6 | Yes | |
HKSZLNNOFSGOKW
|
7.9 | Kd | 408 | — | |
LVUGPVDXTSJQQD
|
7.9 | IC50 | 13 | Yes | |
UPOHPTDDNIQADZ
|
7.9 | IC50 | 2 | — | |
IVZNWJUHDBLKKT
|
7.9 | IC50 | 2 | — | |
ZHBTZVAVYLOIKW
|
7.9 | IC50 | 11 | Yes | |
NPSXOCPQKKCBFX
|
7.8 | IC50 | 3 | Yes | |
GOLYJKYVHGGVMA
|
7.8 | IC50 | 2 | — | |
IVZNWJUHDBLKKT
|
7.8 | IC50 | 2 | — | |
PNEGWAQERPTPDN
|
7.8 | IC50 | 12 | Yes | |
SEJGTFPOEJWEGG
|
7.8 | Kd | 149 | — | |
XYFPWWZEPKGCCK
|
7.8 | IC50 | 34 | — | |
ZCWXCBKGPJOAFQ
|
7.8 | IC50 | 13 | — | |
GNIYUURCQFKRCB
|
7.8 | IC50 | 11 | Yes | |
HTEUQPWFMDGLKN
|
7.8 | IC50 | 6 | Yes | |
FRKWMLCUONAHJH
|
7.8 | IC50 | 13 | Yes | |
KUUKOPMICNKRGE
|
7.8 | IC50 | 12 | Yes |