Target Details
| UniProt AC | P08631 |
|---|---|
| Gene Symbol | HCK |
| Protein Name | Tyrosine-protein kinase HCK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 379
- Clinical molecules 191
- Avg pChEMBL 7.22
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (379)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PHXJVRSECIGDHY
|
10.0 | IC50 | 59 | — | |
UDUPSRWUDACGIS
|
9.7 | IC50 | 13 | Yes | |
ZBNZXTGUTAYRHI
|
9.5 | Kd | 102 | Yes | |
FDVSOQRNTAPCHB
|
9.4 | IC50 | 8 | Yes | |
DKZHIEIQEWZOOJ
|
9.2 | IC50 | 2 | — | |
GXNMERWJFXJFEZ
|
9.2 | IC50 | 2 | — | |
XNHMUNZOELOQNO
|
9.1 | IC50 | 2 | — | |
SSDFTYWIYVWCIE
|
9.0 | IC50 | 17 | — | |
TXXJOMXTCSPSFF
|
8.8 | IC50 | 2 | — | |
REFXTMLPVWSINW
|
8.7 | IC50 | 2 | — | |
JIFZZVZROIFPKB
|
8.7 | IC50 | 5 | — | |
WFRLFWGASBLYTC
|
8.7 | IC50 | 15 | Yes | |
ZBTLTVIYBHYEHL
|
8.7 | IC50 | 13 | Yes | |
ZTQOHJNXDAUMOA
|
8.7 | IC50 | 13 | Yes | |
FDGQFGYDZLTUBK
|
8.6 | IC50 | 2 | — | |
GZOONDJISKPFEJ
|
8.6 | IC50 | 4 | — | |
LYADGAGFYYXXIO
|
8.6 | IC50 | 82 | — | |
FJCORFQIRVXPCY
|
8.5 | IC50 | 4 | — | |
GRFBNEAPKLWFPA
|
8.5 | IC50 | 4 | — | |
GWOFQUMBWYKHFL
|
8.5 | IC50 | 5 | — | |
KIPZYDCBLYBUMY
|
8.5 | IC50 | 4 | — | |
MIAZWLXBNITBFW
|
8.5 | IC50 | 4 | — | |
PDQILYUWWBSUJV
|
8.5 | IC50 | 4 | — | |
SMWGCUOXWXYZPF
|
8.5 | IC50 | 5 | — | |
XJBQSGXAJXTXAC
|
8.5 | IC50 | 5 | — | |
YHVHYWYQEFELOW
|
8.5 | IC50 | 44 | — | |
VAARYSWULJUGST
|
8.5 | Kd | 119 | Yes | |
UBPYILGKFZZVDX
|
8.5 | Kd | 130 | Yes | |
LCYSSHSIKSARGO
|
8.4 | IC50 | 19 | — | |
BBDYTNGLQLQTOV
|
8.4 | IC50 | 4 | — | |
FEFIXEMJIYHFAZ
|
8.4 | IC50 | 4 | — | |
FPSYUXXLCHMFRU
|
8.4 | IC50 | 4 | — | |
IFLRTIBATNZOEH
|
8.4 | IC50 | 4 | — | |
SSIFHFIRVJXKOP
|
8.4 | IC50 | 4 | — | |
UUDAKQZBMTXFJA
|
8.4 | IC50 | 4 | — | |
XHMUIKSUZGOOPZ
|
8.4 | IC50 | 2 | — | |
ZLMVXCGWUJXFNP
|
8.4 | IC50 | 15 | Yes | |
UPOHPTDDNIQADZ
|
8.4 | IC50 | 2 | — | |
QDGTXHCHKQBECZ
|
8.4 | IC50 | 2 | — | |
IWGLXKVBQSBQMC
|
8.4 | IC50 | 13 | Yes | |
PQRFMBAACAPZPP
|
8.3 | IC50 | 12 | Yes | |
AVUUHIYJPTWYNX
|
8.3 | Kd | 9 | — | |
HKSZLNNOFSGOKW
|
8.3 | Ki | 118 | — | |
HYEOMJSVLMONGY
|
8.3 | IC50 | 4 | — | |
PBBRWFOVCUAONR
|
8.3 | IC50 | 26 | Yes | |
QAKIGHBHPHZCJC
|
8.3 | IC50 | 4 | — | |
SXEJPJAKKSSHHC
|
8.3 | IC50 | 4 | — | |
YMXZIONZPMRKQD
|
8.3 | IC50 | 5 | — | |
ZSAJPWOGVMFXHN
|
8.3 | IC50 | 10 | Yes | |
BTIKYUUNPGWLNG
|
8.3 | IC50 | 12 | Yes |