Target Details
UniProt ACP08588
Gene SymbolADRB1
Protein NameBeta-1 adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 541
  • Clinical molecules 2
  • Avg pChEMBL 7.0
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (541)
InChIKey pChEMBL Type Targets Clinical
GPFBLKJURPGHRB 6.4 Kd 3
IHESCUFUOPLPNI 6.4 Ki 2
KUXZXMUDNXFJNC 6.4 Kd 3
LLFZUKMTOZHVQK 6.4 Ki 3
NMTNMGBESHYBOM 6.4 Ki 3
REYSXKCQMOFODI 6.4 IC50 2
YACSDLMXVJCBGL 6.4 Kd 3
YLVVPHSFBDIKPJ 6.4 Ki 2
QAECXSGXRBCERJ 6.3 Ki 2
QXTKUULGJYJUIB 6.3 Ki 3
LWQUXBBBSYMOPD 6.3 Kd 3
NDJLTYJJCSTDDO 6.3 Ki 3
CYUHKBWENYTWOZ 6.3 Kd 3
MTCMWLZKYJYVBZ 6.3 Kd 6
TYQULXNTIHTDSG 6.3 IC50 2
GKTQBPYMIGXPKG 6.3 Ki 21 Yes
GKTQBPYMIGXPKG 6.3 Ki 18
HPTKHKFFMSMJTM 6.3 Ki 3
VBSMKEQICRNWJO 6.3 Ki 2
WATLMDUSELNTHD 6.3 Ki 3
ZATHFADCCIHSFX 6.3 IC50 2
ZQWNZUAMWNPQGR 6.3 Ki 2
GRSIQKKNSPHJED 6.3 Ki 3
MQFHXEQEGSZSEX 6.3 Kd 3
GFNHPWSZFRJUOF 6.3 Kd 3
KMAYGCQZUYYMPJ 6.3 Kd 3
WQRHGJVXZGJYHH 6.3 IC50 2
WRRASIKGHQTERO 6.3 Kd 3
ZLXIUIBLWYKVOG 6.3 IC50 3
VMAXOLZYDATUED 6.3 IC50 2
XSDXBRNBCVMTEE 6.3 Kd 3
YMOLTQUYGLBVRU 6.3 IC50 2
CXWOTFGJCKJHPO 6.3 Ki 2
QTRGGBVZQYMUBP 6.3 IC50 2
XSKNMWQZATUMBK 6.3 IC50 2
AMRDNKZCKDKZFE 6.3 Kd 3
BHBSSMZKXOFWQY 6.2 Ki 3
CXWUYJQOIVNRTF 6.2 Kd 3
FAPFLIWIGPTUPT 6.2 Ki 3
NMEBDKVGJXBMMG 6.2 Kd 3
WKKDUGLKYGNMOU 6.2 Kd 3
CSYYTSAKDHLJGH 6.2 Kd 3
SNWNTDPDTKRCGC 6.2 IC50 2
YDMLHIJQHJTIRS 6.2 Ki 3
YGMWKTPSQYSKCR 6.2 IC50 2
BOHFHHWJKIJTBC 6.2 IC50 2
MDPGYFIGIJWUFG 6.2 Ki 2
OBMZAQJWOSAVBZ 6.2 IC50 2
OZVBMTJYIDMWIL 6.2 Ki 20
QOYHHIBFXOOADH 6.2 Ki 16
2D structure