Target Details
| UniProt AC | P08588 |
|---|---|
| Gene Symbol | ADRB1 |
| Protein Name | Beta-1 adrenergic receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 541
- Clinical molecules 2
- Avg pChEMBL 7.0
KEGG Pathways (13)
- Adrenergic signaling in cardiomyocytes
- Calcium signaling pathway
- Chemical carcinogenesis - receptor activation
- Dilated cardiomyopathy
- Gap junction
- Hormone signaling
- Neuroactive ligand signaling
- Neuroactive ligand-receptor interaction
- Regulation of lipolysis in adipocytes
- Renin secretion
- Salivary secretion
- cAMP signaling pathway
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (541)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QABNYJAOJSVFTR
|
6.1 | IC50 | 2 | — | |
ZWLKZIOYRNEGOR
|
6.1 | IC50 | 2 | — | |
ZMSCROSNCXBMOP
|
6.1 | IC50 | 2 | — | |
QCKDOONRRZRSPO
|
6.0 | IC50 | 2 | — | |
SUROPEFKPIJNCD
|
6.0 | IC50 | 2 | — | |
WBTMIQSFAXDMPJ
|
6.0 | IC50 | 2 | — | |
BNDBBYINHFCCSQ
|
6.0 | IC50 | 2 | — | |
QLHQVTPMIQWMSN
|
6.0 | IC50 | 2 | — | |
SLNOTSHFPJYLEY
|
6.0 | Ki | 2 | — | |
LBELPNBKSBOXOB
|
6.0 | Ki | 3 | — | |
YMJNZSRXRGBYCR
|
6.0 | IC50 | 2 | — | |
AXDLDTSPXTUODG
|
6.0 | Ki | 3 | — | |
LUBDEAGTLSVIAU
|
6.0 | IC50 | 2 | — | |
UPWFWUGEOVNJIM
|
6.0 | IC50 | 2 | — | |
URPKPLOGQTWZLC
|
6.0 | IC50 | 2 | — | |
AOOSJYIINXVNHV
|
6.0 | Ki | 16 | — | |
BVMFDIYNCISFGG
|
6.0 | IC50 | 2 | — | |
CJYLMYWVSLAUFF
|
6.0 | IC50 | 2 | — | |
CNMFEYUJQSQUBJ
|
6.0 | IC50 | 2 | — | |
FUQCILPMICPJAL
|
6.0 | IC50 | 2 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — | |
JKCIKWIXDFDPQX
|
6.0 | IC50 | 2 | — | |
KAALXKXXWZCFLC
|
6.0 | IC50 | 2 | — | |
LWLTZYDRRSELFO
|
6.0 | IC50 | 2 | — | |
MSOUIIHPMJCUNI
|
6.0 | IC50 | 4 | — | |
MXPUBPBHIUDTJX
|
6.0 | Ki | 3 | — | |
NCXAJNHFWXKRON
|
6.0 | IC50 | 2 | — | |
NYBQQHJGLBCUBL
|
6.0 | Ki | 5 | — | |
PCRICIUMMKDSIF
|
6.0 | IC50 | 3 | — | |
PSQPNBVYTLBESR
|
6.0 | IC50 | 2 | — | |
QEQLUORAGYDGGJ
|
6.0 | IC50 | 2 | — | |
RLSSPMNVYVVRQN
|
6.0 | IC50 | 2 | — | |
SVSGFMKNOJDYEE
|
6.0 | IC50 | 2 | — | |
VRJJALQQBINJCH
|
6.0 | IC50 | 2 | — | |
WQMUWTUKVXWONB
|
6.0 | IC50 | 2 | — | |
WWPYNKRNJNPFSG
|
6.0 | IC50 | 2 | — | |
XBRQEMWJALNPLR
|
6.0 | IC50 | 2 | — | |
YCMOYOHTIKWGSW
|
6.0 | Ki | 3 | — | |
YHSGEKJDOIPDMT
|
6.0 | IC50 | 2 | — | |
ZFZUYTCCHMWWTD
|
6.0 | Ki | 9 | — | |
ZUEYCYIOCSMNPN
|
6.0 | Kd | 3 | — |