Target Details
UniProt ACP08588
Gene SymbolADRB1
Protein NameBeta-1 adrenergic receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 541
  • Clinical molecules 2
  • Avg pChEMBL 7.0
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (541)
InChIKey pChEMBL Type Targets Clinical
RBSGUQYXRDKPAE 10.6 Ki 2
GWAMGWDJCYIREE 10.1 Kd 20
IWBMAAUPHUCYCI 10.1 Kd 20
MODBIBJHAWXYOZ 10.1 Kd 20
ZRQMUCDHVVOENY 10.1 Kd 17
SBAJMOUEQDPSIH 10.0 Ki 3
BHIAIPWSVYSKJS 9.7 Ki 2
QHLGXPUIUKSADT 9.6 Ki 6
UMQUQWCJKFOUGV 9.6 Ki 2
NXQMNKUGGYNLBY 9.4 Kd 2
OGHNVEJMJSYVRP 9.3 Ki 18
JZQKKSLKJUAGIC 9.2 IC50 4
TXOCLBKURYXNCG 9.1 Ki 3
QTWVYUJFBIVOHT 9.1 Ki 2
DBHPVKNFKBKJCE 9.0 Kd 2
XSVDIPPEZOQKGV 9.0 Ki 3
GKJZEKSHCJELPL 8.9 Kd 2
HTLWRKRZKFAAAH 8.9 Kd 2
MKYUDVKGSDGIOZ 8.8 Ki 2
STUBIVXIKVVAJL 8.8 Ki 2
UMQUQWCJKFOUGV 8.8 Kd 3
BZWPLBUXCWTALE 8.8 Ki 2
QBHWFJABBIHHGB 8.8 Kd 2
GTTZQULJQRNNER 8.7 Ki 2
SXHDWOIPFGGJDK 8.7 Ki 2
FCMXOBKPGZCHAZ 8.7 Ki 2
XXPNWYXHQVWMTB 8.7 IC50 4
JZQKKSLKJUAGIC 8.7 Ki 5
NBTZMFMFCAFRPY 8.6 IC50 2
PITGAFMHSKTZOO 8.6 Ki 3
AQHHHDLHHXJYJD 8.6 Kd 11
AQHHHDLHHXJYJD 8.6 Ki 11
IMCUOTHFJIPMIY 8.5 Kd 2
HQIRNZOQPUAHHV 8.5 Kd 3
FMJYIEYLOQSTQE 8.5 IC50 2
GYVPBQWEZRVOPO 8.5 Ki 3
XYORPFAZUCCVPS 8.5 Kd 3
GWTZHGSOVZFFPA 8.4 Ki 2
KRCTVIVPCMLXBB 8.4 IC50 2
PCVCNAZGPOOIQN 8.4 Kd 3
FCTFPNMRTWZMQN 8.4 IC50 2
OMKRQXYKQXMQEL 8.4 Ki 3
VAKUOBVYGMAXIO 8.4 IC50 3
VVKYQWBTLQUEAT 8.3 IC50 2
YUDVGSONQUSBKH 8.3 Kd 3
PAZJSJFMUHDSTF 8.3 IC50 4
IXHBTMCLRNMKHZ 8.3 IC50 4
BLJRIMJGRPQVNF 8.3 Ki 4
PAZJSJFMUHDSTF 8.3 IC50 3
SPZVYNXXPJLBRR 8.3 Ki 3
2D structure