Target Details
| UniProt AC | P08581 |
|---|---|
| Gene Symbol | MET |
| Protein Name | Hepatocyte growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF01437 (PSI) PF01403 (Sema) PF01833 (TIG) |
Summary
- Multi-target molecules 1,125
- Clinical molecules 162
- Avg pChEMBL 7.37
KEGG Pathways (25)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Chemical carcinogenesis - reactive oxygen species
- EGFR tyrosine kinase inhibitor resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Focal adhesion
- Gastric cancer
- Hepatocellular carcinoma
- Integrin signaling
- MAPK signaling pathway
- Malaria
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Renal cell carcinoma
- Transcriptional misregulation in cancer
Associated Diseases (8)
Active Molecules (1,125)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SFSRAXHDYDSSCN
|
7.7 | IC50 | 2 | — | |
XZDKAVSSXNBWNJ
|
7.7 | pIC50 | 5 | Yes | |
JJGHHJJQQHUAGN
|
7.7 | IC50 | 2 | — | |
VKBFHTIUXUCYRQ
|
7.7 | Ki | 66 | — | |
BPDPKBWIXIMZMC
|
7.6 | pIC50 | 2 | Yes | |
FCLVBOUURHAHBG
|
7.6 | IC50 | 2 | — | |
IMUUEXXPJMRNER
|
7.6 | IC50 | 2 | — | |
JGJNYXBFXRDVDI
|
7.6 | IC50 | 2 | — | |
LCKSLCUQDDPKQN
|
7.6 | IC50 | 2 | — | |
OIOZTIQUNWLFQV
|
7.6 | IC50 | 3 | — | |
XKPVANIUEZWDCZ
|
7.6 | IC50 | 2 | — | |
XMKAFTZMVDNUII
|
7.6 | IC50 | 2 | — | |
BWXISLRRARTIGU
|
7.6 | IC50 | 6 | — | |
CKICLAQXACKROI
|
7.6 | IC50 | 2 | — | |
JHTHXZUWKNWHSN
|
7.6 | IC50 | 2 | — | |
NWDBTPCKVPWWCM
|
7.6 | IC50 | 2 | — | |
QOMGQLZYIUPQLG
|
7.6 | IC50 | 7 | — | |
VYMTUJBEYOVPCB
|
7.6 | IC50 | 2 | — | |
XMKAFTZMVDNUII
|
7.6 | IC50 | 2 | — | |
OLZPYOIWNSDNMX
|
7.6 | IC50 | 2 | — | |
AWKVKBJHESFTRA
|
7.6 | IC50 | 2 | — | |
BSSQWRSSNZFRMM
|
7.6 | pIC50 | 2 | Yes | |
GGJPKPHOWZDYAP
|
7.6 | IC50 | 2 | — | |
HPBXBZWZAPICIM
|
7.6 | IC50 | 2 | — | |
HTYQIJDCGZYOPT
|
7.6 | IC50 | 2 | — | |
OKCKAUVUVCQSOI
|
7.6 | IC50 | 2 | — | |
DNRDWKZUFWVTKE
|
7.6 | IC50 | 2 | — | |
RKFUKWHBZZWJNX
|
7.6 | pIC50 | 4 | Yes | |
UFAGKVVNSAVENQ
|
7.6 | IC50 | 2 | — | |
BFSZDJBZPXCQJS
|
7.6 | IC50 | 2 | — | |
RKTKWXXUXXANFZ
|
7.6 | IC50 | 2 | — | |
WWFWWACWIOTPBI
|
7.6 | IC50 | 2 | — | |
BXVHRRLJGZKCBN
|
7.6 | IC50 | 2 | — | |
LCCBBQQRBMWQEO
|
7.6 | IC50 | 2 | — | |
HLYLVLPUVNOQHH
|
7.6 | IC50 | 3 | — | |
LZSOTYFDFVIEGI
|
7.6 | IC50 | 4 | — | |
OZIZRJFBDUUQNT
|
7.5 | IC50 | 3 | — | |
RRMOGJHBHWYMHX
|
7.5 | pIC50 | 2 | Yes | |
FERXSPCVEYOEDT
|
7.5 | IC50 | 2 | — | |
RKOUKZKFCAOXCG
|
7.5 | IC50 | 2 | — | |
WIXBTAOMGMZCEY
|
7.5 | IC50 | 2 | — | |
YRCHYHRCBXNYNU
|
7.5 | IC50 | 13 | — | |
ABXAHAOCSWBNBG
|
7.5 | pIC50 | 2 | Yes | |
IKWXNXBFSIAXJW
|
7.5 | IC50 | 2 | — | |
JWQRJKUZDUQDNX
|
7.5 | IC50 | 3 | — | |
RXXOBMLZTZLIBG
|
7.5 | IC50 | 2 | — | |
SGYCGPMBUWGLHB
|
7.5 | IC50 | 2 | — | |
SUYDWRHGHAJQHG
|
7.5 | pIC50 | 2 | Yes | |
VVCJSJLTDUKFKI
|
7.5 | pIC50 | 2 | Yes | |
DWSUPVLNYBTFKY
|
7.5 | IC50 | 2 | — |