Target Details
| UniProt AC | P08581 |
|---|---|
| Gene Symbol | MET |
| Protein Name | Hepatocyte growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF01437 (PSI) PF01403 (Sema) PF01833 (TIG) |
Summary
- Multi-target molecules 1,125
- Clinical molecules 162
- Avg pChEMBL 7.37
KEGG Pathways (25)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Chemical carcinogenesis - reactive oxygen species
- EGFR tyrosine kinase inhibitor resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Focal adhesion
- Gastric cancer
- Hepatocellular carcinoma
- Integrin signaling
- MAPK signaling pathway
- Malaria
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Renal cell carcinoma
- Transcriptional misregulation in cancer
Associated Diseases (8)
Active Molecules (1,125)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JUTMYSXKSLZJQM
|
7.9 | IC50 | 2 | — | |
WWYZAHWIUVISIK
|
7.9 | IC50 | 2 | — | |
BLMPKINHBQAHPE
|
7.9 | IC50 | 2 | — | |
BVGDAZBTIVRTGO
|
7.9 | IC50 | 2 | — | |
BWSKRLZWHCNHLB
|
7.9 | IC50 | 2 | — | |
HLDBRFJDIQDEFJ
|
7.9 | IC50 | 2 | — | |
OWFXKTOLFUQPDJ
|
7.9 | Ki | 36 | — | |
RJZDECGDCKOHBV
|
7.9 | Ki | 70 | — | |
XHORJSJFHVABEA
|
7.9 | Ki | 49 | — | |
JNVFMMAYSXTMTJ
|
7.9 | IC50 | 2 | — | |
XHYQGPMEHCDPLG
|
7.9 | pIC50 | 2 | Yes | |
FWXODUHNWANOFN
|
7.9 | IC50 | 3 | — | |
JFNLWZOMZWJCEF
|
7.9 | IC50 | 2 | — | |
LBFSRNMRNQGAAI
|
7.9 | IC50 | 3 | — | |
MVIYVVFPRORRFN
|
7.9 | IC50 | 2 | — | |
VOMZTXKSRXWVTR
|
7.9 | IC50 | 2 | — | |
YHVAWTSFRPAMNQ
|
7.9 | IC50 | 2 | — | |
ILHJPMFRERKMAB
|
7.9 | IC50 | 2 | — | |
CRQMAEDPCQSZBK
|
7.8 | pIC50 | 2 | Yes | |
DPMQHTABGLRCQK
|
7.8 | IC50 | 5 | — | |
DUTNABYDBFVZOA
|
7.8 | IC50 | 3 | — | |
HBCLIMFCYITYLF
|
7.8 | IC50 | 2 | — | |
LQVXSNNAFNGRAH
|
7.8 | IC50 | 33 | Yes | |
NXLXVWKXBAWMDC
|
7.8 | pIC50 | 2 | Yes | |
PYGNUGPDMKZMBH
|
7.8 | IC50 | 2 | — | |
UQRCJCNVNUFYDX
|
7.8 | IC50 | 27 | — | |
YUOGCICHWDJBLS
|
7.8 | IC50 | 2 | — | |
GGJPKPHOWZDYAP
|
7.8 | IC50 | 2 | — | |
HAFZQSVDZNBXHX
|
7.8 | IC50 | 2 | — | |
NBAROHPFFUMFNW
|
7.8 | IC50 | 3 | — | |
WVNAHDJJLIHTPX
|
7.8 | IC50 | 2 | — | |
GZVQZLVAKXRTHU
|
7.8 | IC50 | 7 | — | |
IZZAJZCFAZXNDC
|
7.8 | pIC50 | 6 | Yes | |
KTEIFNKAUNYNJU
|
7.8 | Ki | 48 | — | |
LNAOKRMVGJXRHU
|
7.8 | IC50 | 2 | — | |
NJCUQMYNSWUWGU
|
7.8 | pIC50 | 2 | Yes | |
QVLIPUSWOSVZPQ
|
7.8 | pIC50 | 2 | Yes | |
WZJWUFBHESGOMB
|
7.8 | IC50 | 2 | — | |
ZQWLWUNEDJXZGN
|
7.8 | IC50 | 2 | — | |
GFIFMJWBJIGJFQ
|
7.8 | IC50 | 2 | — | |
ADLPKFFMGIJZIM
|
7.8 | Ki | 44 | — | |
CVGZRGTXRASJJB
|
7.8 | pIC50 | 2 | Yes | |
OBVABXWHTLZJKU
|
7.8 | IC50 | 2 | — | |
WEHWZYPLPHDXQC
|
7.8 | IC50 | 2 | — | |
IVPRXQPVSHRZHS
|
7.8 | IC50 | 2 | — | |
JEDCUDZEGIOLNY
|
7.8 | Ki | 2 | — | |
MRFFMALERXPRTF
|
7.8 | IC50 | 2 | — | |
YPAMIZOFVIMUOZ
|
7.8 | IC50 | 2 | — | |
FHFKMBKXODPUFW
|
7.8 | IC50 | 5 | — | |
HZQKNWJBZJKRAT
|
7.8 | IC50 | 2 | — |