Target Details
| UniProt AC | P08581 |
|---|---|
| Gene Symbol | MET |
| Protein Name | Hepatocyte growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF01437 (PSI) PF01403 (Sema) PF01833 (TIG) |
Summary
- Multi-target molecules 1,125
- Clinical molecules 162
- Avg pChEMBL 7.37
KEGG Pathways (25)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Chemical carcinogenesis - reactive oxygen species
- EGFR tyrosine kinase inhibitor resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Focal adhesion
- Gastric cancer
- Hepatocellular carcinoma
- Integrin signaling
- MAPK signaling pathway
- Malaria
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Renal cell carcinoma
- Transcriptional misregulation in cancer
Associated Diseases (8)
Active Molecules (1,125)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AKBLFCHEFXTDBF
|
8.2 | IC50 | 2 | — | |
AKBLFCHEFXTDBF
|
8.2 | IC50 | 2 | — | |
HBJCTXQIDBQUKL
|
8.2 | IC50 | 2 | — | |
HVQXOMBEMKJVOC
|
8.2 | IC50 | 2 | — | |
QAXSZRIWQDFFMT
|
8.2 | IC50 | 2 | — | |
AAYNQFQFLVLOHH
|
8.2 | IC50 | 2 | — | |
OEZOMMSDHODKOJ
|
8.2 | IC50 | 2 | — | |
NKVYDBNTELEPBO
|
8.2 | IC50 | 2 | — | |
SEERCQIVLBZZJL
|
8.2 | IC50 | 2 | — | |
AHNSCZJRLJXRAM
|
8.2 | IC50 | 2 | — | |
LDRHWDNTNFXKEE
|
8.2 | IC50 | 3 | — | |
SQYNPZYBHGTSOY
|
8.2 | IC50 | 5 | — | |
AXFCKENUDNTMRB
|
8.2 | IC50 | 2 | — | |
CKRJSIFFXMHDSE
|
8.2 | pIC50 | 3 | Yes | |
DGVPNVQBSCWKJG
|
8.2 | IC50 | 2 | — | |
GTDCAFNNNVCDJN
|
8.2 | pIC50 | 2 | Yes | |
HTZHPXKKPOLGTR
|
8.2 | IC50 | 9 | — | |
LOLPPWBBNUVNQZ
|
8.2 | Kd | 97 | Yes | |
NNVFVZWTQYUWJO
|
8.2 | IC50 | 2 | — | |
NXVHOYBQFPQTBF
|
8.2 | IC50 | 3 | — | |
ZSXQYYKWSXJOSG
|
8.2 | pIC50 | 2 | Yes | |
ZXWBEPIEIMDBRM
|
8.2 | pIC50 | 4 | Yes | |
DWUNWBPFOCBLPR
|
8.1 | IC50 | 2 | — | |
GFLLLFKVJIGOGF
|
8.1 | IC50 | 2 | — | |
XYJHFAIWNWCPJD
|
8.1 | IC50 | 2 | — | |
DGRCFAYRKDYEMX
|
8.1 | IC50 | 7 | — | |
JKOLVOLGJWWVFD
|
8.1 | IC50 | 2 | — | |
VUWNSIKRZRWGIE
|
8.1 | IC50 | 2 | — | |
QPYYLLKCTPKJEO
|
8.1 | IC50 | 3 | — | |
RYQBKVFFHMNFTM
|
8.1 | IC50 | 3 | — | |
FERXSPCVEYOEDT
|
8.1 | IC50 | 4 | — | |
JHZOJILVCGEIFB
|
8.1 | IC50 | 3 | — | |
AEAOPPHJQXFHPG
|
8.1 | IC50 | 2 | — | |
AROMUEFGOQGFHF
|
8.1 | IC50 | 3 | — | |
GEZKQLDGHARZBQ
|
8.1 | IC50 | 2 | — | |
HBNFTDDTRWSQBS
|
8.1 | pIC50 | 2 | Yes | |
MCCCQFAOMZMZKE
|
8.1 | Ki | 52 | — | |
MWVKLRSIDOXBSE
|
8.1 | IC50 | 4 | — | |
OEUQPIPNLAICFE
|
8.1 | pIC50 | 3 | Yes | |
QMNCWLZBRSTKTL
|
8.1 | IC50 | 2 | — | |
RFMLRIANOITTIG
|
8.1 | IC50 | 2 | — | |
RGNHKJWHFIPHIM
|
8.1 | Ki | 66 | — | |
WOBLFEIWTSKVMT
|
8.1 | pIC50 | 2 | Yes | |
YWDRXTGAHCQDDT
|
8.1 | IC50 | 2 | — | |
ZCCJKVBTHCOISJ
|
8.1 | Ki | 46 | — | |
BBZWMCIWNJHTMG
|
8.1 | IC50 | 2 | — | |
FDHGNGABRSFZEF
|
8.1 | IC50 | 2 | — | |
VCMSULGORSGFSP
|
8.1 | IC50 | 3 | — | |
VZNJIFQUJWERJH
|
8.1 | IC50 | 2 | — | |
NKVYDBNTELEPBO
|
8.1 | IC50 | 2 | — |