Target Details
| UniProt AC | P08581 |
|---|---|
| Gene Symbol | MET |
| Protein Name | Hepatocyte growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF01437 (PSI) PF01403 (Sema) PF01833 (TIG) |
Summary
- Multi-target molecules 1,125
- Clinical molecules 162
- Avg pChEMBL 7.37
KEGG Pathways (25)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Chemical carcinogenesis - reactive oxygen species
- EGFR tyrosine kinase inhibitor resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Focal adhesion
- Gastric cancer
- Hepatocellular carcinoma
- Integrin signaling
- MAPK signaling pathway
- Malaria
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Renal cell carcinoma
- Transcriptional misregulation in cancer
Associated Diseases (8)
Active Molecules (1,125)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YHVHYWYQEFELOW
|
8.4 | IC50 | 44 | — | |
YYPVGQBXTJNGFW
|
8.4 | IC50 | 4 | — | |
DAOGGCDCTXWDAX
|
8.4 | IC50 | 2 | — | |
FGPIVIJULBNRBX
|
8.4 | IC50 | 4 | — | |
XEPIWGLSVOVBHX
|
8.4 | IC50 | 2 | — | |
CTSDMCNSBRVZGJ
|
8.4 | IC50 | 7 | — | |
ABXVJDAAJIHQCN
|
8.4 | IC50 | 2 | — | |
AIDASDNWZFQVSE
|
8.4 | IC50 | 2 | — | |
LDXRJMINDNMMRX
|
8.3 | IC50 | 3 | — | |
BUKHWHCWUHMPKB
|
8.3 | IC50 | 3 | — | |
BZWHAJVPFKNIQF
|
8.3 | IC50 | 3 | — | |
PLODQYLMGYEBRS
|
8.3 | IC50 | 2 | — | |
QHADVLVFMKEIIP
|
8.3 | IC50 | 9 | — | |
IZUHPEAVOSEXHO
|
8.3 | IC50 | 2 | — | |
LZHNGGOUJMOCJB
|
8.3 | IC50 | 2 | — | |
OFPQHQDWNLXNKV
|
8.3 | IC50 | 2 | — | |
OSKAWGHRJOWPNQ
|
8.3 | IC50 | 2 | — | |
XYDNMOZJKOGZLS
|
8.3 | IC50 | 2 | — | |
LWVKBWDPQJMBIE
|
8.3 | IC50 | 2 | — | |
ONSZEUCTVQJHOZ
|
8.3 | IC50 | 9 | — | |
FVKQINCBAYQVHF
|
8.3 | IC50 | 2 | — | |
SMKGLAAOEUNWFQ
|
8.3 | IC50 | 2 | — | |
WBEVSLNQXYPTEA
|
8.3 | pIC50 | 2 | Yes | |
WQROZMCEHXFGBY
|
8.3 | IC50 | 2 | — | |
YEICXZQUNLMHNW
|
8.3 | pIC50 | 2 | Yes | |
AHTUGEFRTOJHHF
|
8.3 | IC50 | 2 | — | |
QSFGBNSTSAEDNQ
|
8.3 | IC50 | 2 | — | |
GLHCZNFHZBSVML
|
8.3 | IC50 | 2 | — | |
HVQXOMBEMKJVOC
|
8.3 | IC50 | 2 | — | |
GHRAGOBMSUDFEQ
|
8.3 | IC50 | 2 | — | |
VVGBSNRZVJGQFL
|
8.3 | IC50 | 5 | — | |
NNYPTMWKSXSUEP
|
8.3 | IC50 | 2 | — | |
GYCPBMYHPVDKFK
|
8.2 | IC50 | 3 | — | |
KHSXMHYXEDTYDH
|
8.2 | IC50 | 2 | — | |
QKQBOUUDOCRITG
|
8.2 | IC50 | 2 | — | |
RYZPDFHBMIKLBP
|
8.2 | IC50 | 2 | — | |
DGMFNZXEGKFREH
|
8.2 | IC50 | 2 | — | |
JQKLADMYWZPROY
|
8.2 | IC50 | 2 | — | |
NXHDXFKJDNLGQF
|
8.2 | pIC50 | 2 | Yes | |
QHIKHPOSGIFPMN
|
8.2 | pIC50 | 2 | Yes | |
UFICVEHDQUKCEA
|
8.2 | pIC50 | 4 | Yes | |
WCHXVWBCCCSTPJ
|
8.2 | pIC50 | 2 | Yes | |
BSFOFLYNEZXJRV
|
8.2 | IC50 | 2 | — | |
DMUUMPYJFUHKCR
|
8.2 | IC50 | 2 | — | |
GCVRKWYNRILXKN
|
8.2 | IC50 | 2 | — | |
QMILKASSWHCTOF
|
8.2 | IC50 | 4 | — | |
QYCCMZVRTHGSBB
|
8.2 | IC50 | 2 | — | |
SOZIDKBTBOAWJZ
|
8.2 | IC50 | 2 | — | |
UNVJKMKVJXWKNX
|
8.2 | IC50 | 2 | — | |
AEKJPCHGTMQXDQ
|
8.2 | IC50 | 2 | — |