Target Details
| UniProt AC | P08581 |
|---|---|
| Gene Symbol | MET |
| Protein Name | Hepatocyte growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF01437 (PSI) PF01403 (Sema) PF01833 (TIG) |
Summary
- Multi-target molecules 1,125
- Clinical molecules 162
- Avg pChEMBL 7.37
KEGG Pathways (25)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Chemical carcinogenesis - reactive oxygen species
- EGFR tyrosine kinase inhibitor resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Focal adhesion
- Gastric cancer
- Hepatocellular carcinoma
- Integrin signaling
- MAPK signaling pathway
- Malaria
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Renal cell carcinoma
- Transcriptional misregulation in cancer
Associated Diseases (8)
Active Molecules (1,125)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GEGCXGMFUYJULA
|
6.3 | Ki | 30 | Yes | |
GJOXRIYWDHESDF
|
6.3 | Ki | 27 | — | |
HCNIBOQWDVOZKF
|
6.3 | Ki | 26 | — | |
HZPACYSNLOCDLW
|
6.3 | Ki | 48 | — | |
IAKGNUWZPSPEKU
|
6.3 | Ki | 19 | — | |
KRIUNPBAQZGFQA
|
6.3 | Ki | 76 | — | |
KUDLEBZUOBVRGB
|
6.3 | IC50 | 2 | — | |
NECQZMQPXFYVOY
|
6.3 | Ki | 26 | — | |
PROLIXHVRCJEFH
|
6.3 | Ki | 46 | — | |
SFPWNTQWFFNJIH
|
6.3 | Ki | 48 | — | |
XMGFTZYNTYNOOJ
|
6.3 | Ki | 10 | — | |
DKNUPRMJNUQNHR
|
6.3 | Kd | 33 | — | |
GRWMCJDUSSENHT
|
6.3 | IC50 | 2 | — | |
WZSFRCWKHKFQMG
|
6.3 | IC50 | 2 | — | |
MJMQNGOVXMCDGQ
|
6.3 | IC50 | 2 | — | |
BAKDYDIANXRUHQ
|
6.3 | IC50 | 3 | — | |
SVZJDNDOMDBENZ
|
6.3 | IC50 | 2 | — | |
AEDKPHMRPYJLGA
|
6.3 | IC50 | 2 | — | |
BAGLRIYGLUAGSG
|
6.3 | IC50 | 3 | — | |
BEBIQNBKDFRLBS
|
6.3 | IC50 | 2 | — | |
BSMUSWHXZAXDID
|
6.3 | IC50 | 3 | — | |
CSMSPOIEMWPZLD
|
6.3 | IC50 | 2 | — | |
DIHBLMSEOXGIKG
|
6.3 | IC50 | 2 | — | |
DTKKTUUDABIULF
|
6.3 | IC50 | 3 | — | |
GAMIOFOGSQTZLB
|
6.3 | IC50 | 2 | — | |
HBENISDMECHQSQ
|
6.3 | IC50 | 3 | — | |
HYHPUWFUFKIZPE
|
6.3 | IC50 | 2 | — | |
JGXXVRONABNGOX
|
6.3 | IC50 | 2 | — | |
JTGIOGAVFYKHHY
|
6.3 | IC50 | 2 | — | |
JTNXTIPDQKHRDT
|
6.3 | IC50 | 3 | — | |
JTNXTIPDQKHRDT
|
6.3 | IC50 | 3 | — | |
KKJZILBNEHLFLH
|
6.3 | IC50 | 2 | — | |
LIHDGASTMHTMGG
|
6.3 | IC50 | 2 | — | |
MYUJBDVTLXXMHN
|
6.3 | IC50 | 3 | — | |
NAHDXRNJVZITKJ
|
6.3 | IC50 | 2 | — | |
OSAMADCNPNUCEI
|
6.3 | IC50 | 2 | — | |
OTXJGYRNPGIHAP
|
6.3 | IC50 | 3 | — | |
QKLHJJJNGDFUIT
|
6.3 | IC50 | 3 | — | |
QLICCXIUWDZMJX
|
6.3 | IC50 | 3 | — | |
RAPKAHFDNKOYTF
|
6.3 | IC50 | 3 | — | |
RMERCRTVGVRYLB
|
6.3 | IC50 | 2 | — | |
SHBAHISDWOTLDJ
|
6.3 | IC50 | 2 | — | |
SKIWKGOSDXYROV
|
6.3 | IC50 | 2 | — | |
SPMVMDHWKHCIDT
|
6.3 | IC50 | 30 | — | |
SUCTWUOQZPDKSP
|
6.3 | IC50 | 2 | — | |
TXZRIDXMQZUDMK
|
6.3 | IC50 | 3 | — | |
UJNNBNJYUJMGSK
|
6.3 | IC50 | 2 | — | |
UZSBNRYHYVACAH
|
6.3 | IC50 | 2 | — | |
YBCVPFLUANOFHV
|
6.3 | IC50 | 3 | — | |
ZSDIFSIINICKHA
|
6.3 | IC50 | 2 | — |