Target Details
| UniProt AC | P08581 |
|---|---|
| Gene Symbol | MET |
| Protein Name | Hepatocyte growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF01437 (PSI) PF01403 (Sema) PF01833 (TIG) |
Summary
- Multi-target molecules 1,125
- Clinical molecules 162
- Avg pChEMBL 7.37
KEGG Pathways (25)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Chemical carcinogenesis - reactive oxygen species
- EGFR tyrosine kinase inhibitor resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Focal adhesion
- Gastric cancer
- Hepatocellular carcinoma
- Integrin signaling
- MAPK signaling pathway
- Malaria
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Renal cell carcinoma
- Transcriptional misregulation in cancer
Associated Diseases (8)
Active Molecules (1,125)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HBQMROYUNHRFSB
|
8.9 | IC50 | 5 | — | |
KAPOJQHBFXHFOU
|
8.9 | IC50 | 2 | — | |
OHLUERTUZNIQEE
|
8.9 | IC50 | 3 | — | |
OJDVWGXCETZZLV
|
8.9 | IC50 | 2 | — | |
BYYYCNUDMZSOGS
|
8.9 | pIC50 | 5 | Yes | |
GIGLKJOCNUGOJM
|
8.9 | IC50 | 2 | — | |
GZMFYPWWSXGVTC
|
8.9 | IC50 | 2 | — | |
HSAQBRJGYZIVJP
|
8.9 | pIC50 | 5 | Yes | |
YEGSATWQBXVWBX
|
8.9 | IC50 | 6 | — | |
PSTHAQGLUUIJDB
|
8.8 | IC50 | 6 | — | |
PSTHAQGLUUIJDB
|
8.8 | IC50 | 4 | — | |
UFYWONKSWCXKNY
|
8.8 | IC50 | 5 | — | |
CXQUSKUCZSYVLJ
|
8.8 | IC50 | 2 | — | |
ZMTGUZWATGQQFE
|
8.8 | IC50 | 2 | — | |
IBISBIYLXKDMHL
|
8.8 | IC50 | 2 | — | |
XVKMYLMSWNIAHF
|
8.8 | IC50 | 2 | — | |
MWXLURJNASFGGM
|
8.8 | IC50 | 5 | — | |
OPWIMESOOZSXGC
|
8.8 | IC50 | 2 | — | |
WDAHGVLBPINGHW
|
8.8 | IC50 | 6 | — | |
CXQHYVUVSFXTMY
|
8.8 | IC50 | 154 | — | |
PDYXPCKITKHFOZ
|
8.8 | IC50 | 2 | — | |
ULHLSSWDQFLSBL
|
8.8 | IC50 | 6 | — | |
VKRRGKOVGYHCBL
|
8.8 | IC50 | 2 | — | |
YIFMGCJQLZYTAA
|
8.8 | IC50 | 2 | — | |
ZEQSGOFKTMWPAI
|
8.8 | IC50 | 2 | — | |
OBSFXHDOLBYWRJ
|
8.7 | pIC50 | 7 | Yes | |
QCSPHKYKAODHGS
|
8.7 | IC50 | 3 | — | |
DQVUCDBOFDTXMU
|
8.7 | IC50 | 5 | — | |
IBUOCLLDDGZTCA
|
8.7 | IC50 | 2 | — | |
IXULLLZCNUKGBJ
|
8.7 | IC50 | 6 | — | |
UUDQJODJTHYBOX
|
8.7 | IC50 | 2 | — | |
WXOGYBWIHWKUMA
|
8.7 | IC50 | 2 | — | |
BRXZUOJFGVQTAB
|
8.7 | pIC50 | 3 | Yes | |
GLBZSOQDAOLMGC
|
8.7 | Ki | 23 | Yes | |
ILVXQVHFMCJXTE
|
8.7 | IC50 | 2 | — | |
LKUSYUYBQDJFNA
|
8.7 | IC50 | 2 | — | |
OPMJBWVXRQIVBZ
|
8.7 | IC50 | 8 | — | |
XDXHFPNTAVKXEG
|
8.7 | IC50 | 2 | — | |
OZXPSVBSQRGYFB
|
8.7 | IC50 | 2 | — | |
WUIOBNGTWSVFMF
|
8.7 | IC50 | 2 | — | |
HXGIQMKSZVMZAD
|
8.7 | IC50 | 2 | — | |
JYBQEMYHVMILOJ
|
8.7 | IC50 | 5 | — | |
KEDANNMRCOENMZ
|
8.7 | IC50 | 7 | — | |
AAYNQFQFLVLOHH
|
8.6 | IC50 | 2 | — | |
MVAYPHGEGDDSJN
|
8.6 | IC50 | 6 | — | |
ABKGHWKSGAOXGR
|
8.6 | IC50 | 2 | — | |
LODWOBAYUQRWKD
|
8.6 | IC50 | 7 | — | |
MGUCSMZMGMTIOE
|
8.6 | IC50 | 2 | — | |
UMMZZOSIEGYDTO
|
8.6 | Kd | 2 | — | |
FVPYEAORCOKOLV
|
8.6 | IC50 | 6 | — |