Target Details
| UniProt AC | P08581 |
|---|---|
| Gene Symbol | MET |
| Protein Name | Hepatocyte growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF01437 (PSI) PF01403 (Sema) PF01833 (TIG) |
Summary
- Multi-target molecules 1,125
- Clinical molecules 162
- Avg pChEMBL 7.37
KEGG Pathways (25)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Chemical carcinogenesis - reactive oxygen species
- EGFR tyrosine kinase inhibitor resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Focal adhesion
- Gastric cancer
- Hepatocellular carcinoma
- Integrin signaling
- MAPK signaling pathway
- Malaria
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Renal cell carcinoma
- Transcriptional misregulation in cancer
Associated Diseases (8)
Active Molecules (1,125)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FVUINRBQOUDLSO
|
6.7 | IC50 | 2 | — | |
UMBIRSZUCJNBHB
|
6.7 | IC50 | 18 | — | |
AEUQVUHYNJZUMV
|
6.7 | Kd | 2 | — | |
ALCCHVWXJSBREH
|
6.7 | IC50 | 2 | — | |
CBUSZPVAZDIGMN
|
6.7 | IC50 | 2 | — | |
DVRROHBOBHXFEN
|
6.7 | IC50 | 2 | — | |
FGQUZTPOBIQTMT
|
6.7 | IC50 | 2 | — | |
FOSNOEXXSOQKEV
|
6.7 | IC50 | 2 | — | |
FQYLJBVSYHZWLT
|
6.7 | Ki | 35 | Yes | |
GCBJDOWIQHMCMR
|
6.7 | Ki | 84 | — | |
GCYXEGSPUDSZJY
|
6.7 | Ki | 82 | — | |
GDATVDHFQFRHKH
|
6.7 | IC50 | 2 | — | |
GQTGXSGWXVDRDZ
|
6.7 | IC50 | 2 | — | |
GYJDQSJMOWWHIN
|
6.7 | IC50 | 2 | — | |
IELXVRGBXDSTMS
|
6.7 | IC50 | 2 | — | |
IPEDTKUJEWGEIY
|
6.7 | IC50 | 2 | — | |
JCWYTIFWSKODPB
|
6.7 | IC50 | 2 | — | |
JHYHWHUTTXJICB
|
6.7 | Ki | 18 | — | |
JJKGYGMFHAYASJ
|
6.7 | IC50 | 3 | — | |
JLYICKALDOGPTC
|
6.7 | IC50 | 2 | — | |
KQCHFNHYSYAEPM
|
6.7 | IC50 | 2 | — | |
LBFFPDPAHKPYNJ
|
6.7 | IC50 | 2 | — | |
MIEQOSSLRLYSHP
|
6.7 | IC50 | 2 | — | |
NRFIMGFSYNRJEZ
|
6.7 | IC50 | 2 | — | |
PGUNHFIEAZPDMH
|
6.7 | IC50 | 2 | — | |
PSXWVEYYLHUUMT
|
6.7 | IC50 | 2 | — | |
QWVYEFCLRGZMJR
|
6.7 | pIC50 | 2 | Yes | |
RNZVSXPOBSLRDN
|
6.7 | IC50 | 2 | — | |
UYJNQQDJUOUFQJ
|
6.7 | Ki | 68 | — | |
WUIZHOHGGZBREA
|
6.7 | IC50 | 2 | — | |
XVUGJMRSDJSHFU
|
6.7 | IC50 | 2 | — | |
YYPKOMNJRZRWIC
|
6.7 | Ki | 26 | — | |
CKVXYSBVFGGCGL
|
6.7 | IC50 | 5 | — | |
UAWDRWOANYZGFE
|
6.7 | IC50 | 2 | — | |
AOICHKUMZOVLSN
|
6.7 | IC50 | 2 | — | |
MFYBSISLMUXOGK
|
6.7 | IC50 | 2 | — | |
RBGSTRWPZHSCTD
|
6.7 | IC50 | 2 | — | |
UXBXTSWBNHTFRX
|
6.7 | pIC50 | 3 | Yes | |
YYLKKYCXAOBSRM
|
6.7 | Kd | 191 | — | |
GJEWUZOGSANRGN
|
6.7 | IC50 | 2 | — | |
QWSBWFZCNLMQCF
|
6.7 | IC50 | 2 | — | |
SSPYHBZSDDTSFN
|
6.7 | IC50 | 9 | — | |
RFKWZWJQRQCLJF
|
6.7 | IC50 | 2 | — | |
STKCTXOVMCUJSB
|
6.7 | IC50 | 4 | — | |
BHMWKIPRPJDXFD
|
6.6 | IC50 | 2 | — | |
KNWKQGFTYAADHZ
|
6.6 | IC50 | 2 | — | |
VBFGYZJIKZDDLS
|
6.6 | IC50 | 2 | — | |
DOHXUBMMYMAIQP
|
6.6 | IC50 | 2 | — | |
HHKOKFHTWVYTJK
|
6.6 | IC50 | 4 | — | |
DVRMYRDLCLUXQP
|
6.6 | IC50 | 2 | — |