Target Details
| UniProt AC | P08581 |
|---|---|
| Gene Symbol | MET |
| Protein Name | Hepatocyte growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF01437 (PSI) PF01403 (Sema) PF01833 (TIG) |
Summary
- Multi-target molecules 1,125
- Clinical molecules 162
- Avg pChEMBL 7.37
KEGG Pathways (25)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Chemical carcinogenesis - reactive oxygen species
- EGFR tyrosine kinase inhibitor resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Focal adhesion
- Gastric cancer
- Hepatocellular carcinoma
- Integrin signaling
- MAPK signaling pathway
- Malaria
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Renal cell carcinoma
- Transcriptional misregulation in cancer
Associated Diseases (8)
Active Molecules (1,125)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BSKHIANLHIEMMY
|
7.3 | IC50 | 3 | — | |
CCLHDMIHAHKLKJ
|
7.3 | IC50 | 2 | — | |
CLNZOVOBAXNFGG
|
7.3 | IC50 | 3 | — | |
CPRQKIQZMBAYGL
|
7.3 | IC50 | 3 | — | |
CQACOGKETKCZSQ
|
7.3 | IC50 | 2 | — | |
CRAHFBSLWSAFHP
|
7.3 | IC50 | 3 | — | |
CRZSZRSFXGWQFK
|
7.3 | IC50 | 2 | — | |
DVYRJIORBQLTKB
|
7.3 | IC50 | 2 | — | |
FJPDSDCACJWODZ
|
7.3 | IC50 | 2 | — | |
FKCWHHYUMFGOPY
|
7.3 | IC50 | 2 | — | |
FWCRQKIZZVMWID
|
7.3 | IC50 | 2 | — | |
GBGXUVPPNWEOLE
|
7.3 | IC50 | 3 | — | |
GTVNQWNESMCZOI
|
7.3 | IC50 | 2 | — | |
GVMBNRTYQPUNMR
|
7.3 | IC50 | 2 | — | |
HBBJPARWIXBJRM
|
7.3 | IC50 | 2 | — | |
HHJPYGDVCUQLTQ
|
7.3 | IC50 | 2 | — | |
IGPWVRHOMPPQQD
|
7.3 | IC50 | 2 | — | |
IHDYOFLXCUAKSS
|
7.3 | IC50 | 2 | — | |
IHFWPQZJKNTETJ
|
7.3 | IC50 | 2 | — | |
ILARUASUFRIPAV
|
7.3 | IC50 | 2 | — | |
IOLSMTRHLGQZQC
|
7.3 | IC50 | 2 | — | |
IQPXOYXEBLLUIP
|
7.3 | IC50 | 2 | — | |
IVZFDQZKNNXELU
|
7.3 | IC50 | 2 | — | |
JLPWQBJIMNSJND
|
7.3 | IC50 | 2 | — | |
JMQFGWVOJUJDJC
|
7.3 | IC50 | 2 | — | |
JMXLDWRDBOMQJR
|
7.3 | IC50 | 2 | — | |
JRNKDLIGAZRRAU
|
7.3 | IC50 | 2 | — | |
KBIAXSIBSRAFPH
|
7.3 | IC50 | 2 | — | |
KIGCBVALXFPNSJ
|
7.3 | IC50 | 2 | — | |
KOGINFSZWQZUSG
|
7.3 | IC50 | 3 | — | |
KVOQWZUWKAIRLV
|
7.3 | IC50 | 2 | — | |
LAFVEBGIXOWENG
|
7.3 | IC50 | 2 | — | |
LAKJAOFXTCJILU
|
7.3 | IC50 | 2 | — | |
LCSVZVBSNJJXAP
|
7.3 | IC50 | 2 | — | |
LGJITSYEXZMUHA
|
7.3 | IC50 | 2 | — | |
LSDQPXYSLVYYIB
|
7.3 | IC50 | 2 | — | |
LSEVBZSAGKKXQF
|
7.3 | IC50 | 2 | — | |
LVYXERPKYAQGKM
|
7.3 | IC50 | 4 | — | |
MBRAXNBBJZZVAE
|
7.3 | IC50 | 2 | — | |
MCIVTOPWKOAUNP
|
7.3 | IC50 | 2 | — | |
MIDVZIJNTYYCGV
|
7.3 | IC50 | 2 | — | |
NPUDQTABBPAVEO
|
7.3 | IC50 | 2 | — | |
NQYRQYRTPHFSEO
|
7.3 | IC50 | 3 | — | |
NYDHCFXFFOGARN
|
7.3 | IC50 | 2 | — | |
OACZVJRZOXXBDJ
|
7.3 | IC50 | 3 | — | |
OADZCVZONHKWGC
|
7.3 | IC50 | 2 | — | |
OERZGXZCWQGXSB
|
7.3 | IC50 | 2 | — | |
OGJOGSMHNSGUML
|
7.3 | IC50 | 2 | — | |
OKXRAGPSTORXAZ
|
7.3 | IC50 | 3 | — | |
OTKTYQXOBFJYGG
|
7.3 | IC50 | 3 | — |