Target Details
| UniProt AC | P08581 |
|---|---|
| Gene Symbol | MET |
| Protein Name | Hepatocyte growth factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF01437 (PSI) PF01403 (Sema) PF01833 (TIG) |
Summary
- Multi-target molecules 1,125
- Clinical molecules 162
- Avg pChEMBL 7.37
KEGG Pathways (25)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- Chemical carcinogenesis - reactive oxygen species
- EGFR tyrosine kinase inhibitor resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Focal adhesion
- Gastric cancer
- Hepatocellular carcinoma
- Integrin signaling
- MAPK signaling pathway
- Malaria
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Renal cell carcinoma
- Transcriptional misregulation in cancer
Associated Diseases (8)
Active Molecules (1,125)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FUNHEVBLXUQXLG
|
7.5 | IC50 | 2 | — | |
LEJSTVMXRPKNQA
|
7.5 | IC50 | 2 | — | |
LFKPJUFFMOTFRX
|
7.5 | IC50 | 6 | — | |
RBKXLMGSZLUVAU
|
7.5 | pIC50 | 2 | Yes | |
MHCPAORAYMTGCZ
|
7.5 | Ki | 37 | — | |
MNUPLQVJAOMLAS
|
7.5 | IC50 | 2 | — | |
NPKHYQHLPSZNHP
|
7.5 | IC50 | 2 | — | |
ORRNXRYWGDUDOG
|
7.5 | IC50 | 5 | — | |
OWRXHGAFWZFFCW
|
7.5 | Ki | 113 | — | |
RYYNGWLOYLRZLK
|
7.5 | Ki | 104 | — | |
VUPKYIDSZYTBHB
|
7.5 | IC50 | 2 | — | |
GJTGIHCBLUARCQ
|
7.5 | IC50 | 2 | — | |
NDECJXFIPXCRJU
|
7.5 | pIC50 | 2 | Yes | |
QJKRRPUDVWORKT
|
7.5 | IC50 | 2 | — | |
QUNNUMNERCPGKL
|
7.5 | pIC50 | 2 | Yes | |
BRFFOZKQXZVVQO
|
7.5 | IC50 | 2 | — | |
DVYVSTMPCPXIIT
|
7.5 | IC50 | 2 | — | |
HDVHNQRHFIRVBQ
|
7.5 | IC50 | 2 | — | |
HQHYTWCENUFKDZ
|
7.5 | IC50 | 2 | — | |
ICYMRJXTNSDJCF
|
7.5 | IC50 | 2 | — | |
KMSULJIFXXDZAE
|
7.5 | IC50 | 2 | — | |
ONYDOUQLFUMDET
|
7.5 | IC50 | 2 | — | |
STZMYLKPKCSIEC
|
7.5 | IC50 | 2 | — | |
WABZCKCXZGRTFB
|
7.5 | IC50 | 2 | — | |
WKZAFJWEZVPGCZ
|
7.5 | IC50 | 2 | — | |
ANDWXAGCNLNBJR
|
7.5 | IC50 | 2 | — | |
YYFOSKNQHFIIIM
|
7.5 | IC50 | 2 | — | |
MTBUICNMPXYSAM
|
7.5 | IC50 | 2 | — | |
SOBJVDFONGAIIH
|
7.5 | IC50 | 2 | — | |
DPDFZTKJHYCDSX
|
7.4 | IC50 | 3 | — | |
JSDFIHRUQVWHKK
|
7.4 | IC50 | 2 | — | |
KTQKHIKEYBROHW
|
7.4 | IC50 | 2 | — | |
VLYCWERLMYAMSM
|
7.4 | IC50 | 2 | — | |
ZOEMYGXYNBNGJA
|
7.4 | IC50 | 2 | — | |
JZMKNOWKNYJUOM
|
7.4 | IC50 | 3 | — | |
PZDZBMUDLPDHQV
|
7.4 | IC50 | 2 | — | |
QDDUFIFVBIXXSF
|
7.4 | IC50 | 2 | — | |
QXGDVAINKPZMRY
|
7.4 | IC50 | 2 | — | |
IKPJWGNTDNCFPS
|
7.4 | IC50 | 3 | — | |
IYUWNROPEIAYPD
|
7.4 | IC50 | 2 | — | |
RDOUYNQAILJAAS
|
7.4 | IC50 | 2 | — | |
VRFBKBFDZDKNBO
|
7.4 | IC50 | 2 | — | |
WKIJVZYIYLQZNN
|
7.4 | IC50 | 2 | — | |
BIKYDWLMTPRSQL
|
7.4 | Ki | 50 | — | |
CAHIYUNFMZWRQZ
|
7.4 | IC50 | 2 | — | |
DJNWXYTWORPJNI
|
7.4 | pIC50 | 3 | Yes | |
FIODPWXACNUFML
|
7.4 | IC50 | 2 | — | |
FLEAYYMORDPWAJ
|
7.4 | Ki | 90 | — | |
LOYACYJWFBZPCW
|
7.4 | IC50 | 3 | — | |
OZHHLHNBHBGTSP
|
7.4 | pIC50 | 3 | Yes |