Target Details
| UniProt AC | P08514 |
|---|---|
| Gene Symbol | ITGA2B |
| Protein Name | Integrin alpha-IIb |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,322
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- Neutrophil extracellular trap formation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Platelet activation
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Small cell lung cancer
Associated Diseases (4)
Active Molecules (1,322)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QEUNDODSNWYTBN
|
7.8 | IC50 | 2 | — | |
RFWCQGQYCWHAEC
|
7.8 | IC50 | 2 | — | |
SAFNKDHVPKIPDD
|
7.8 | IC50 | 2 | — | |
VITFKBICHMWBSD
|
7.8 | IC50 | 2 | — | |
VNNMTZFLPCRBMP
|
7.8 | IC50 | 2 | — | |
IFUROQAKNZUNFY
|
7.8 | IC50 | 5 | — | |
AKOSSGWXDCGWFL
|
7.8 | IC50 | 4 | — | |
ALIJPZPRXMWHRP
|
7.8 | IC50 | 2 | — | |
HBIADZKHMCJYMA
|
7.8 | IC50 | 2 | — | |
QVMQHOLQYLDBQM
|
7.8 | IC50 | 2 | — | |
RVIXCVCUEFSALD
|
7.8 | IC50 | 2 | — | |
TXXFSQAOZCGSGM
|
7.8 | IC50 | 2 | — | |
UYKFRSOVXIPIKF
|
7.8 | IC50 | 2 | — | |
MNSHWMCGPFNHKK
|
7.8 | IC50 | 3 | — | |
DKGATRXTJTUOON
|
7.8 | IC50 | 3 | — | |
GYDZTZMAFRCBOY
|
7.8 | IC50 | 2 | — | |
HPSQGYXTQFSXQR
|
7.8 | IC50 | 3 | — | |
HTPRMRASPJUHGG
|
7.8 | IC50 | 3 | — | |
LWHWQLNSWIQIMG
|
7.8 | IC50 | 4 | — | |
MHVOJKFXMPOUON
|
7.8 | IC50 | 2 | — | |
NHGBKPGAKQVOMR
|
7.8 | IC50 | 2 | — | |
PXSDSRKJCWOYNE
|
7.8 | IC50 | 2 | — | |
ZWFZEAWYCOFELN
|
7.8 | IC50 | 2 | — | |
WTSKVLROSCOUMY
|
7.8 | IC50 | 2 | — | |
GKOZTPMILPOVDI
|
7.8 | IC50 | 2 | — | |
IJQHTEYCWOTDQL
|
7.8 | IC50 | 2 | — | |
ZNBYKEFOMOGFQE
|
7.8 | IC50 | 2 | — | |
AKHLJKBUPDHNIH
|
7.7 | IC50 | 2 | — | |
BYAJINXSXQREIN
|
7.7 | IC50 | 2 | — | |
CBELHQKPOFWOOH
|
7.7 | IC50 | 2 | — | |
IWAXDMYAVCCIQY
|
7.7 | IC50 | 2 | — | |
MQWGOPKAWPNVQO
|
7.7 | IC50 | 2 | — | |
MVIVEASLSGRCJF
|
7.7 | IC50 | 2 | — | |
OKEKRFLAQTYOCR
|
7.7 | IC50 | 3 | — | |
RWFZWACTJSUZOO
|
7.7 | IC50 | 2 | — | |
XIWNZCZUNRLAND
|
7.7 | IC50 | 2 | — | |
YUDGHBDJGIBNNN
|
7.7 | IC50 | 2 | — | |
CRIVUOYMMLIKDM
|
7.7 | Kd | 2 | — | |
GJTFLSXWEKTYAH
|
7.7 | IC50 | 2 | — | |
POQNQXDDMZDMDU
|
7.7 | IC50 | 2 | — | |
ULFCJKOYMHZEGE
|
7.7 | Ki | 2 | — | |
FPWWHFZBMPQJMS
|
7.7 | IC50 | 3 | — | |
ACHJOQIILIANHB
|
7.7 | IC50 | 4 | — | |
BDHMASHCRICMNC
|
7.7 | IC50 | 2 | — | |
BQTUWUXJPAYSPB
|
7.7 | IC50 | 2 | — | |
CNSWTCWKTAAVJS
|
7.7 | IC50 | 2 | — | |
DYXWODXGLWRHBW
|
7.7 | IC50 | 2 | — | |
FLYVHWZXQKAHIV
|
7.7 | IC50 | 2 | — | |
HKTFAZNSYXVZNN
|
7.7 | IC50 | 2 | — | |
IREXQQUAADPBFC
|
7.7 | Ki | 2 | — |