Target Details
| UniProt AC | P08514 |
|---|---|
| Gene Symbol | ITGA2B |
| Protein Name | Integrin alpha-IIb |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,322
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- Neutrophil extracellular trap formation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Platelet activation
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Small cell lung cancer
Associated Diseases (4)
Active Molecules (1,322)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DMXRDQJVBMEHPP
|
7.9 | IC50 | 2 | — | |
FWUBZVPKPDMTEU
|
7.9 | IC50 | 2 | — | |
GVYNMUHOCJCTAC
|
7.9 | IC50 | 3 | — | |
HUKZLLZKJKIAFJ
|
7.9 | Kd | 2 | — | |
ISSFWLVXRAXPAT
|
7.9 | IC50 | 2 | — | |
KXTBADBGYGMUFO
|
7.9 | IC50 | 2 | — | |
NCRTXTOOWLTIEL
|
7.9 | IC50 | 3 | — | |
PAFICDQSPQMTGA
|
7.9 | IC50 | 2 | — | |
PNKDBLJVPXRVTK
|
7.9 | Kd | 2 | — | |
ZQPJXQFVXFPVOP
|
7.9 | IC50 | 2 | — | |
YTPVKTLAFFSGBR
|
7.9 | IC50 | 3 | — | |
ZWFZEAWYCOFELN
|
7.9 | IC50 | 2 | — | |
CFKZYRJYUHWTIW
|
7.9 | IC50 | 2 | — | |
CSICLXCUTLXRPU
|
7.9 | Kd | 2 | — | |
DWUDTTQIPXVNRZ
|
7.9 | IC50 | 2 | — | |
FMQLAOUMABGLDL
|
7.9 | IC50 | 2 | — | |
HLIQBOMFPPBSKB
|
7.9 | IC50 | 2 | — | |
KBBXMNQBVKMYCZ
|
7.9 | IC50 | 4 | — | |
KTHYBTKKKGIYPR
|
7.9 | Kd | 2 | — | |
MVCBOXJOFRGFIR
|
7.9 | IC50 | 2 | — | |
GPYDNKNVGLPQHE
|
7.9 | IC50 | 2 | — | |
SRLJDTUHNPUPHU
|
7.9 | IC50 | 2 | — | |
DYYSGNJUTBUSGU
|
7.9 | IC50 | 2 | — | |
KRAZOLZZRSRPAE
|
7.9 | IC50 | 4 | — | |
POPLTANACXUDAZ
|
7.9 | IC50 | 2 | — | |
QTVKUFZTCJLGEJ
|
7.9 | IC50 | 2 | — | |
PTBOFZKNVXEWSK
|
7.9 | Ki | 2 | — | |
UDFNVENGUDURFM
|
7.9 | IC50 | 2 | — | |
CRBNIXMHJDLKNC
|
7.8 | IC50 | 2 | — | |
CWDMXFFPROLWHT
|
7.8 | IC50 | 2 | — | |
DSEQSPZXYSBJIV
|
7.8 | IC50 | 2 | — | |
FOIPXCGYGBYXAS
|
7.8 | IC50 | 5 | — | |
JQVNOQWITDASST
|
7.8 | IC50 | 2 | — | |
LTIDGEKEJCQKNB
|
7.8 | IC50 | 2 | — | |
NXKFHFCWTSGLDC
|
7.8 | IC50 | 4 | — | |
OUYHRBRXZUOZRC
|
7.8 | IC50 | 4 | — | |
PECKOTHCSJMAES
|
7.8 | IC50 | 2 | — | |
QDBNJVOFTDUTIW
|
7.8 | IC50 | 2 | — | |
XQXXKDXHJWWTMY
|
7.8 | IC50 | 2 | — | |
DIMDWQUSJSWNOO
|
7.8 | IC50 | 5 | — | |
VWSBHFWKGOESTL
|
7.8 | IC50 | 2 | — | |
WGHKPKSITIVVNZ
|
7.8 | IC50 | 2 | — | |
BOHIOMJEXMWHQC
|
7.8 | IC50 | 2 | — | |
DMJMBJHEDODVMW
|
7.8 | IC50 | 3 | — | |
HXYXRRMFBLDLDJ
|
7.8 | Kd | 2 | — | |
KOSFSUYNKQIHHY
|
7.8 | IC50 | 2 | — | |
LONYGERIAVPFRY
|
7.8 | IC50 | 2 | — | |
NDJRYOZGPUGFQI
|
7.8 | IC50 | 2 | — | |
NDJZSISKTPMXEV
|
7.8 | Kd | 2 | — | |
OPSRUAAFZJIVQO
|
7.8 | IC50 | 2 | — |