Target Details
| UniProt AC | P08514 |
|---|---|
| Gene Symbol | ITGA2B |
| Protein Name | Integrin alpha-IIb |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,322
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- Neutrophil extracellular trap formation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Platelet activation
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Small cell lung cancer
Associated Diseases (4)
Active Molecules (1,322)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PUFOHCGQIDICBZ
|
8.1 | Kd | 2 | — | |
COKMIXFXJJXBQG
|
8.1 | IC50 | 4 | — | |
CQDWPOURVPAZAM
|
8.1 | IC50 | 5 | — | |
FHHKNJSJONAARK
|
8.1 | IC50 | 2 | — | |
JPXXAQAAXBCQPT
|
8.1 | Kd | 2 | — | |
KSPAZKMCXAMIPC
|
8.1 | IC50 | 3 | — | |
UMBVVGYRMZYGDW
|
8.1 | IC50 | 2 | — | |
YFEFXIJHEGDAHU
|
8.1 | IC50 | 2 | — | |
ZPOXUYJIZHGYGR
|
8.1 | IC50 | 2 | — | |
DDMLNTCTSCHYTO
|
8.0 | IC50 | 2 | — | |
VOZZIKGZFLWFGA
|
8.0 | IC50 | 3 | — | |
UWQLXVUHLJYGKT
|
8.0 | Ki | 2 | — | |
CEKNHWXPXHFXSX
|
8.0 | Ki | 2 | — | |
FCTUEQVODTYVHM
|
8.0 | IC50 | 3 | — | |
RNRNOOHZNNWVAO
|
8.0 | IC50 | 2 | — | |
XMCFUKKHFHSEML
|
8.0 | IC50 | 2 | — | |
LMECSRGVSCMHBF
|
8.0 | IC50 | 2 | — | |
ALDNYPOFXBNJLU
|
8.0 | IC50 | 2 | — | |
BRSXVPVATKZROV
|
8.0 | IC50 | 2 | — | |
BSXTXDDIXVXJQU
|
8.0 | Kd | 2 | — | |
FMXQBVYTEHKMDV
|
8.0 | IC50 | 2 | — | |
JESHEQMKKYQWKH
|
8.0 | IC50 | 4 | — | |
LRRHPVLPULZTFH
|
8.0 | IC50 | 2 | — | |
NKYASGUMKORFAJ
|
8.0 | IC50 | 2 | — | |
SMICYQXKVBGSTO
|
8.0 | IC50 | 2 | — | |
XIFBKSWCVWRQPS
|
8.0 | Ki | 2 | — | |
YINCHOOHNDSILR
|
8.0 | IC50 | 4 | — | |
YUQXUXRQTHCXHR
|
8.0 | IC50 | 2 | — | |
NACYWTUZCONRAO
|
8.0 | IC50 | 2 | — | |
RUZPDEXRJNESMI
|
8.0 | IC50 | 2 | — | |
ULMWVACPLANFSN
|
8.0 | IC50 | 2 | — | |
PACNGEUJCLRLPB
|
8.0 | IC50 | 2 | — | |
BNRNDWNDFOMWFM
|
8.0 | IC50 | 2 | — | |
CZEAWFMLBALEFP
|
8.0 | IC50 | 2 | — | |
KALOYQBAVHVFJS
|
8.0 | IC50 | 5 | — | |
OIHPLUDPXSEGBG
|
8.0 | IC50 | 2 | — | |
SBUMUHUTBKYAPS
|
8.0 | IC50 | 4 | — | |
TZZMWRLTTWMKCL
|
8.0 | IC50 | 2 | — | |
VCYXSHVQNGNXQO
|
8.0 | IC50 | 3 | — | |
VVKBGBCCSDVWHK
|
8.0 | IC50 | 3 | — | |
VXMVUSYMRFXJMC
|
8.0 | IC50 | 2 | — | |
XOBFRYRGVGQXQH
|
8.0 | Kd | 2 | — | |
XOINBHSFUQZGLB
|
8.0 | IC50 | 2 | — | |
ZZXJPZTUZLYRTN
|
8.0 | IC50 | 2 | — | |
CCEWOJIAQCICDN
|
8.0 | IC50 | 2 | — | |
CUNMRDASFORTJM
|
7.9 | IC50 | 2 | — | |
WTSKVLROSCOUMY
|
7.9 | IC50 | 2 | — | |
YWYVDMBBVYVCTP
|
7.9 | IC50 | 2 | — | |
XKFYFSNOQRUIAO
|
7.9 | Kd | 2 | — | |
BXPUXQXIESIGAE
|
7.9 | IC50 | 2 | — |