Target Details
| UniProt AC | P08514 |
|---|---|
| Gene Symbol | ITGA2B |
| Protein Name | Integrin alpha-IIb |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,322
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- Neutrophil extracellular trap formation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Platelet activation
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Small cell lung cancer
Associated Diseases (4)
Active Molecules (1,322)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VZYNONIAPDJFNO
|
8.2 | IC50 | 2 | — | |
LSUARKLZJJZSPC
|
8.2 | Kd | 2 | — | |
MMRLXTCMJMOLTL
|
8.2 | IC50 | 2 | — | |
OFMXNBIPYOLGBH
|
8.2 | IC50 | 3 | — | |
UWKPPOAXIFLKJM
|
8.2 | IC50 | 3 | — | |
XWBPHLLWVDTCSH
|
8.2 | Kd | 2 | — | |
FPKOGTAFKSLZLD
|
8.2 | IC50 | 2 | — | |
WVAHTVNIUCSTBB
|
8.2 | IC50 | 2 | — | |
JWRYVLUXFOYZCH
|
8.2 | IC50 | 2 | — | |
LUAGPVPPCBTVMI
|
8.2 | IC50 | 2 | — | |
PYELMOFQPMMHKM
|
8.2 | IC50 | 3 | — | |
SEJKHYQTPOZVIX
|
8.2 | IC50 | 2 | — | |
UFIWBTUUDZMPRH
|
8.2 | Kd | 2 | — | |
GDEQCJXHHVMPLM
|
8.2 | IC50 | 2 | — | |
GXNRMXKXTHPZDX
|
8.2 | IC50 | 5 | — | |
LSMPPNWISBTMIU
|
8.2 | IC50 | 2 | — | |
LWGPKVXXVDWZFF
|
8.2 | IC50 | 2 | — | |
NACYWTUZCONRAO
|
8.2 | IC50 | 2 | — | |
OKHOVATVMTUXHZ
|
8.2 | IC50 | 2 | — | |
OYCLLPDCZQPWQL
|
8.2 | IC50 | 2 | — | |
WQBFXJCREXXMOQ
|
8.2 | IC50 | 2 | — | |
HNJOHJBYQFWLOL
|
8.1 | IC50 | 2 | — | |
NENWIXCUUFUHIH
|
8.1 | IC50 | 3 | — | |
PYZOVVQJTLOHDG
|
8.1 | IC50 | 2 | — | |
QOZKFVLJGZGBOI
|
8.1 | IC50 | 3 | — | |
WYJONACSFWJWGN
|
8.1 | IC50 | 2 | — | |
MHRXUWQLKAROGA
|
8.1 | Kd | 2 | — | |
IGLOTTSZPFMUAC
|
8.1 | Kd | 2 | — | |
QKICCTXUZWAFQK
|
8.1 | IC50 | 2 | — | |
QMRDCHKQISKMJS
|
8.1 | IC50 | 2 | — | |
VZZBPIKSQGUSRZ
|
8.1 | Kd | 2 | — | |
CGSLGBRMSMBNMX
|
8.1 | IC50 | 6 | — | |
TVTYTTGLAUMQMH
|
8.1 | Kd | 2 | — | |
ALPHCBAGUUJBBU
|
8.1 | IC50 | 2 | — | |
GXXMLWSLPOFULG
|
8.1 | IC50 | 2 | — | |
MBNNZQMWRRSBHP
|
8.1 | IC50 | 2 | — | |
NCDMAEGCMKJPAZ
|
8.1 | IC50 | 2 | — | |
RMPDPJUTEPDOAS
|
8.1 | IC50 | 2 | — | |
UHHDYMXTEYGGTM
|
8.1 | Ki | 2 | — | |
XBGMACJUNQNMBD
|
8.1 | Ki | 3 | — | |
XJCXTPBGVGQFQE
|
8.1 | IC50 | 2 | — | |
YNBHAPKHWDNTMZ
|
8.1 | IC50 | 2 | — | |
FAUWCTMBSRSLQY
|
8.1 | IC50 | 2 | — | |
KMXIJCGQJFYWTC
|
8.1 | IC50 | 2 | — | |
KCZDQEZSAWQHPZ
|
8.1 | IC50 | 2 | — | |
AQIWTLCCMPNDGQ
|
8.1 | IC50 | 2 | — | |
BHOGTSLQMNCJHA
|
8.1 | IC50 | 2 | — | |
OVXHVHVMKYQQMG
|
8.1 | Ki | 2 | — | |
UCKMCHCSOYXGOJ
|
8.1 | IC50 | 2 | — | |
NPNSEDOLVQCILC
|
8.1 | IC50 | 2 | — |