Target Details
| UniProt AC | P08514 |
|---|---|
| Gene Symbol | ITGA2B |
| Protein Name | Integrin alpha-IIb |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,322
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- Neutrophil extracellular trap formation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Platelet activation
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Small cell lung cancer
Associated Diseases (4)
Active Molecules (1,322)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ULKYPKCVQKXPOK
|
8.4 | IC50 | 2 | — | |
VDCCBVPSQROOHU
|
8.4 | IC50 | 2 | — | |
UIJBJQDAZCEJGM
|
8.4 | IC50 | 2 | — | |
FEURVUPSCVOVSS
|
8.3 | Ki | 2 | — | |
XVJMRPYMUCTESW
|
8.3 | Ki | 2 | — | |
JXRHFSZNVUPMJD
|
8.3 | IC50 | 3 | — | |
PDZPUQQVGSDNOJ
|
8.3 | IC50 | 3 | — | |
UIJBJQDAZCEJGM
|
8.3 | IC50 | 2 | — | |
BNFSEAYFTNCGLP
|
8.3 | IC50 | 2 | — | |
DNYYJQPHMWSUJW
|
8.3 | IC50 | 2 | — | |
IUYFYZYWSXDLLJ
|
8.3 | IC50 | 2 | — | |
JVBMRJFKTRWIIF
|
8.3 | IC50 | 2 | — | |
LFYAXIXLMQDEKZ
|
8.3 | IC50 | 2 | — | |
OCNALRIBAIFGLP
|
8.3 | IC50 | 3 | — | |
RSEPVNVGKQWNDW
|
8.3 | IC50 | 2 | — | |
VYEAVDMFFXTEBM
|
8.3 | IC50 | 2 | — | |
XGDVRXHWQGEVTD
|
8.3 | IC50 | 3 | — | |
ZNGZDOVQBYPJEY
|
8.3 | IC50 | 2 | — | |
NCPUFPHVKAPNOO
|
8.3 | IC50 | 2 | — | |
QQEZTKRLXQSFTL
|
8.3 | Kd | 2 | — | |
ZFSXCHHVEXOSLC
|
8.3 | IC50 | 2 | — | |
BLZOWNLJBLDRTL
|
8.3 | IC50 | 2 | — | |
GEXLWFJEDGQQNS
|
8.3 | IC50 | 2 | — | |
QOZKFVLJGZGBOI
|
8.3 | IC50 | 3 | — | |
UJVHDCIYLCPNMX
|
8.3 | IC50 | 2 | — | |
HWRXVANHVCXVHA
|
8.3 | IC50 | 3 | — | |
KFNHSIQLBWLFMH
|
8.3 | IC50 | 2 | — | |
SFULVLPBMKAKLA
|
8.2 | IC50 | 2 | — | |
NSXMNJVSOKYCEJ
|
8.2 | IC50 | 2 | — | |
QULYZHFZLOZQQS
|
8.2 | IC50 | 2 | — | |
NXTXRLGABIDNIS
|
8.2 | IC50 | 2 | — | |
ADXRXCZYDSDWJG
|
8.2 | IC50 | 2 | — | |
BDFMVIGZRRIXCL
|
8.2 | IC50 | 5 | — | |
FESCEKWSTPKQHV
|
8.2 | IC50 | 2 | — | |
JQQPAMCEEOBVRO
|
8.2 | IC50 | 2 | — | |
KOSZDUGLIZYKDV
|
8.2 | IC50 | 2 | — | |
NOGJEZSRANWTRH
|
8.2 | IC50 | 2 | — | |
NZRIBORZQOXVCV
|
8.2 | Kd | 2 | — | |
PKIIHLJERYMZGK
|
8.2 | IC50 | 2 | — | |
PUXOGOOLLVFISN
|
8.2 | IC50 | 2 | — | |
RCCYAIQAQJPLAH
|
8.2 | IC50 | 3 | — | |
TVZONMAFMCMGKU
|
8.2 | IC50 | 2 | — | |
TZZMWRLTTWMKCL
|
8.2 | IC50 | 2 | — | |
VEXMPESRUXSYPU
|
8.2 | IC50 | 2 | — | |
WVKRQRRDBUVAHI
|
8.2 | IC50 | 2 | — | |
KDXGTKAQPXSESN
|
8.2 | IC50 | 2 | — | |
PQBZVJZWTNXWCX
|
8.2 | Kd | 2 | — | |
VJJPPEQXMGSWDU
|
8.2 | IC50 | 3 | — | |
FBOPIPGFCRATJI
|
8.2 | IC50 | 2 | — | |
SDTYJAQHROYESA
|
8.2 | IC50 | 2 | — |