Target Details
| UniProt AC | P08514 |
|---|---|
| Gene Symbol | ITGA2B |
| Protein Name | Integrin alpha-IIb |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,322
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- Neutrophil extracellular trap formation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Platelet activation
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Small cell lung cancer
Associated Diseases (4)
Active Molecules (1,322)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TYTHBXMTSPUPRQ
|
8.6 | IC50 | 2 | — | |
LKTCUFLNSKQNFZ
|
8.6 | IC50 | 2 | — | |
LQHWNHQINCFOIZ
|
8.6 | IC50 | 2 | — | |
YIJHNENQTDBNGG
|
8.6 | IC50 | 2 | — | |
XSBCDEUAXRNIMC
|
8.6 | IC50 | 2 | — | |
IRAXRQFCCSHQDX
|
8.6 | Kd | 2 | — | |
JUCUUAVAOJAIHU
|
8.6 | Ki | 2 | — | |
YITSCMGHJOGUNC
|
8.6 | Ki | 3 | — | |
KCPZTHQHJHVUCK
|
8.5 | IC50 | 3 | — | |
ONCDSJSLWNCDLA
|
8.5 | IC50 | 2 | — | |
ABNXKGFLZFSILK
|
8.5 | IC50 | 2 | — | |
CQERSJFWLNZCJI
|
8.5 | IC50 | 2 | — | |
GUTGOHPTMQPGTD
|
8.5 | IC50 | 3 | — | |
LOTOEFNCKZSRAC
|
8.5 | IC50 | 2 | — | |
POPLTANACXUDAZ
|
8.5 | IC50 | 2 | — | |
QVTQDWZYXPQJCE
|
8.5 | IC50 | 2 | — | |
RUFGUKZOARQZPD
|
8.5 | Ki | 2 | — | |
RWGBUALVFDFMJM
|
8.5 | IC50 | 2 | — | |
TVMGTJHIWQJZIM
|
8.5 | IC50 | 2 | — | |
WDTHWJIIRVVYRP
|
8.5 | IC50 | 2 | — | |
WIQNHDTZROVWEI
|
8.5 | IC50 | 2 | — | |
WIZNRUGPDHNTSZ
|
8.5 | IC50 | 2 | — | |
WWDVDVKEFFDGFA
|
8.5 | IC50 | 3 | — | |
XKLZVTVODPFBIC
|
8.5 | IC50 | 2 | — | |
XNQTZNPDLAFJJK
|
8.5 | IC50 | 2 | — | |
ZCBCTVUDWUBKKH
|
8.5 | IC50 | 2 | — | |
XKFYFSNOQRUIAO
|
8.5 | Kd | 2 | — | |
CECDTIOXBMVUGI
|
8.5 | Ki | 2 | — | |
BLIAKAQPONHNOO
|
8.5 | IC50 | 2 | — | |
SVHYTSHIZOYMFB
|
8.5 | IC50 | 2 | — | |
XKFYFSNOQRUIAO
|
8.5 | IC50 | 2 | — | |
AJZXCRQRDSKMDW
|
8.5 | Kd | 2 | — | |
SUTFGPKMGSBIER
|
8.5 | Kd | 2 | — | |
HWPUQFFXBNMTKS
|
8.5 | IC50 | 2 | — | |
XGDVRXHWQGEVTD
|
8.5 | IC50 | 3 | — | |
BEIUZYAXIMVQKS
|
8.4 | IC50 | 2 | — | |
FVGFTYFYGPWTIR
|
8.4 | Kd | 2 | — | |
GHKOZFUXJGLMAL
|
8.4 | IC50 | 2 | — | |
TWQKVYIVXPBLEV
|
8.4 | IC50 | 2 | — | |
VHKHAQYPTPVIAP
|
8.4 | IC50 | 3 | — | |
MFGHNUHLUBBJOD
|
8.4 | IC50 | 2 | — | |
NLJFFXADHHBXSL
|
8.4 | IC50 | 2 | — | |
POMPVFVGEMHCEN
|
8.4 | IC50 | 2 | — | |
BCMLZQVZOQFOSL
|
8.4 | IC50 | 2 | — | |
GPKDWNWVODHEAY
|
8.4 | IC50 | 2 | — | |
KXLMLPVYDRIZFO
|
8.4 | IC50 | 2 | — | |
PYZOVVQJTLOHDG
|
8.4 | Ki | 2 | — | |
QOZKFVLJGZGBOI
|
8.4 | IC50 | 2 | — | |
QZSFFLWIZLMTAZ
|
8.4 | IC50 | 2 | — | |
WLRISAYEIGZWPZ
|
8.4 | IC50 | 2 | — |