Target Details
| UniProt AC | P08514 |
|---|---|
| Gene Symbol | ITGA2B |
| Protein Name | Integrin alpha-IIb |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 1,322
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- Neutrophil extracellular trap formation
- PI3K-Akt signaling pathway
- Pathways in cancer
- Platelet activation
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Small cell lung cancer
Associated Diseases (4)
Active Molecules (1,322)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZSMRGIMZBIOFKN
|
11.9 | IC50 | 2 | — | |
BPBHTITUTUZWBT
|
11.2 | IC50 | 3 | — | |
DGSYYUPRYQBSAI
|
10.6 | IC50 | 2 | — | |
WWPKVHRHQNABNG
|
10.6 | IC50 | 3 | — | |
MUWWGBUXCFRNCO
|
10.2 | IC50 | 2 | — | |
FFYHCEWZIRARDA
|
10.1 | IC50 | 2 | — | |
SVESXPIJWQQCBW
|
10.0 | IC50 | 2 | — | |
LOLMVTRGQZKBHS
|
10.0 | IC50 | 2 | — | |
CYKYNQSFAYHHEZ
|
10.0 | IC50 | 2 | — | |
CYKYNQSFAYHHEZ
|
10.0 | IC50 | 3 | — | |
FGJKSKYLEOZELA
|
10.0 | IC50 | 3 | — | |
WHDDGMQNGFSWHS
|
10.0 | IC50 | 2 | — | |
HFXICNGRABOTIL
|
9.9 | IC50 | 2 | — | |
UBJJRHHGGWEKRK
|
9.9 | IC50 | 2 | — | |
BZNWTXRYYZHACY
|
9.9 | IC50 | 2 | — | |
CQHDUHCWSJOZFD
|
9.9 | IC50 | 2 | — | |
QRGILGTYGXRRFJ
|
9.9 | IC50 | 2 | — | |
RFJPNVAPTYAFSN
|
9.9 | IC50 | 2 | — | |
AQNSLCJLLMFYBT
|
9.8 | IC50 | 2 | — | |
XIUUVOUXDREGQI
|
9.8 | IC50 | 2 | — | |
ABNXKGFLZFSILK
|
9.8 | IC50 | 2 | — | |
YSLIZGZENLHKBF
|
9.8 | IC50 | 2 | — | |
MCDJJGKLMCJYFS
|
9.8 | IC50 | 2 | — | |
NKIPTRIPXHQDGW
|
9.8 | IC50 | 6 | — | |
QAFIKBJSAZTLCJ
|
9.8 | IC50 | 2 | — | |
NJHGFLNQVAIERE
|
9.8 | IC50 | 2 | — | |
GFNRURIBKUNSSG
|
9.7 | IC50 | 2 | — | |
NIAUTJLMLQTPHC
|
9.7 | IC50 | 3 | — | |
HAWHNGUKUZPYEE
|
9.7 | IC50 | 4 | — | |
JGWWDWJMZWLSKE
|
9.7 | IC50 | 2 | — | |
BGLLQJHWAUGNSA
|
9.7 | IC50 | 3 | — | |
QZBZOURIVJUOIH
|
9.7 | IC50 | 2 | — | |
ZCBCTVUDWUBKKH
|
9.7 | IC50 | 2 | — | |
AFEBUYQIVROWSL
|
9.7 | IC50 | 2 | — | |
DFDCHFSRONUYME
|
9.6 | IC50 | 2 | — | |
TZYPGXPOZINIRX
|
9.6 | IC50 | 2 | — | |
LOZUMZUMWUTBLC
|
9.6 | IC50 | 2 | — | |
ARJWFIGFOOVYAR
|
9.6 | IC50 | 2 | — | |
IPLLAQOFEDGGKD
|
9.5 | IC50 | 4 | — | |
UQEWVVUNGPKKKR
|
9.5 | IC50 | 6 | — | |
WEXQBLSMARBRMG
|
9.5 | IC50 | 6 | — | |
HDNLLSLLYCIFIU
|
9.5 | IC50 | 2 | — | |
ABNXKGFLZFSILK
|
9.4 | IC50 | 2 | — | |
AJCAJRVJXQOQGR
|
9.4 | IC50 | 2 | — | |
WWWQNOCFIMKBQL
|
9.4 | IC50 | 2 | — | |
FGJKSKYLEOZELA
|
9.4 | IC50 | 2 | — | |
GHKJCEINAARURY
|
9.4 | IC50 | 2 | — | |
JSXUDXGPZPGJOP
|
9.4 | IC50 | 2 | — | |
XQUJDYKAECREGU
|
9.4 | IC50 | 2 | — | |
DVTSXXOIRGTVES
|
9.4 | IC50 | 2 | — |