Target Details
| UniProt AC | P08473 |
|---|---|
| Gene Symbol | MME |
| Protein Name | Neprilysin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01431 (Peptidase_M13) PF05649 (Peptidase_M13_N) |
Summary
- Multi-target molecules 252
- Clinical molecules 3
- Avg pChEMBL 7.77
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (252)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UVFBPEBPXILYRM
|
6.8 | Ki | 3 | — | |
REUFMJWXJQZYAJ
|
6.8 | IC50 | 3 | — | |
AWWVJFGCYBSRKO
|
6.8 | IC50 | 2 | — | |
BNGVWMNLGADUIP
|
6.8 | IC50 | 3 | — | |
VCPVOGSIRZPBGD
|
6.8 | IC50 | 2 | — | |
ZPFSKFCSVXPMBD
|
6.8 | Ki | 6 | Yes | |
KZAYYAIBZWKHEY
|
6.7 | Ki | 2 | — | |
NJJGKDPBXMIWPF
|
6.7 | Ki | 2 | — | |
BROFGMFOFNHCBY
|
6.7 | IC50 | 2 | — | |
DOBNVUFHFMVMDB
|
6.7 | IC50 | 2 | — | |
JIKXDFOHRKWQIU
|
6.7 | Ki | 2 | — | |
OHEMLLQWDPOUER
|
6.7 | IC50 | 3 | — | |
VNEWJBSOCHQZLJ
|
6.7 | Ki | 2 | — | |
QRJBXCBBMUHKDQ
|
6.6 | IC50 | 2 | — | |
RTROYMXMLRVHBZ
|
6.6 | IC50 | 2 | — | |
ITMFWUAKJPURIP
|
6.6 | Ki | 3 | — | |
YCZFGFJXTINBHZ
|
6.6 | IC50 | 2 | — | |
CXDCBPLMHAFCCH
|
6.5 | IC50 | 2 | — | |
IEBMXVZQILSQHG
|
6.5 | IC50 | 3 | — | |
RUTFYHHMLQZRQB
|
6.5 | Ki | 3 | — | |
BXEKJAAOIPQIDR
|
6.5 | IC50 | 2 | — | |
YIFOVNSRCOGRFA
|
6.5 | IC50 | 2 | — | |
IWURQOHGXLKXDJ
|
6.5 | IC50 | 2 | — | |
IXTVKPZUQDUYAH
|
6.5 | IC50 | 2 | — | |
VMBLGPAYYKVWDU
|
6.5 | IC50 | 3 | — | |
ONNUXPTYPGZZBK
|
6.5 | IC50 | 2 | — | |
CHKOUVAKPRIMRS
|
6.4 | IC50 | 2 | — | |
YSFYVNRABGRTNY
|
6.4 | IC50 | 2 | — | |
VHXDFOBQYJQMPJ
|
6.4 | IC50 | 2 | — | |
ZOFFBAOTPKMRBJ
|
6.4 | Ki | 2 | — | |
KLCDUNQMSZJEDY
|
6.3 | IC50 | 2 | — | |
UVUIZZPSNWBCEK
|
6.3 | IC50 | 2 | — | |
VDEOJAQFLHVZHV
|
6.3 | IC50 | 2 | — | |
IXIRWVIYLLRFNN
|
6.3 | IC50 | 2 | — | |
TYXFDFMUHPWCDX
|
6.2 | IC50 | 2 | — | |
QJZUXIPDHISQFZ
|
6.2 | Ki | 2 | — | |
GMDAQACCLFTFJO
|
6.2 | IC50 | 2 | — | |
MAMIBVRNOYOUBU
|
6.2 | IC50 | 2 | — | |
XHAYUYYNXCLCFY
|
6.2 | IC50 | 2 | — | |
CUXSRYOPSIUUQD
|
6.2 | IC50 | 2 | — | |
RBSIIEZEHKNSIW
|
6.2 | Ki | 2 | — | |
BROFGMFOFNHCBY
|
6.2 | IC50 | 2 | — | |
DOBNVUFHFMVMDB
|
6.2 | IC50 | 2 | — | |
BNWWCJCEOOIWCA
|
6.1 | IC50 | 2 | — | |
DMDAAWYUUQFVGJ
|
6.1 | IC50 | 3 | — | |
HBVPPCWYEOLLHL
|
6.1 | IC50 | 2 | — | |
SYACYTRJPUYQOP
|
6.1 | IC50 | 2 | — | |
ICVAKVXFPOSUDK
|
6.0 | IC50 | 3 | — | |
BIWWMKYCSUXSIM
|
6.0 | IC50 | 2 | — | |
OUSUIQLLVUDFMT
|
6.0 | Ki | 3 | — |