Target Details
| UniProt AC | P08473 |
|---|---|
| Gene Symbol | MME |
| Protein Name | Neprilysin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01431 (Peptidase_M13) PF05649 (Peptidase_M13_N) |
Summary
- Multi-target molecules 252
- Clinical molecules 3
- Avg pChEMBL 7.77
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (252)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JRAQIPPUUOUHFM
|
7.5 | Ki | 2 | — | |
POIKHACBOPACCB
|
7.5 | Ki | 2 | — | |
POIKHACBOPACCB
|
7.5 | Ki | 2 | — | |
DRWPQXKJHUNFJS
|
7.4 | IC50 | 2 | — | |
HSJQIQUIXIQNLN
|
7.4 | Ki | 3 | — | |
VVIGQDQMSRGEBC
|
7.4 | IC50 | 3 | — | |
VVPLZIBCVXZTPQ
|
7.4 | Ki | 3 | — | |
QVLBZMKHYLEWGB
|
7.4 | Ki | 2 | — | |
XRWGWRHXWJHKMY
|
7.4 | IC50 | 2 | — | |
YYPVNXPFSJDVAO
|
7.4 | IC50 | 2 | — | |
DOLNCCYFNWYJPI
|
7.3 | Ki | 3 | — | |
CVTQKTZYWUYCJJ
|
7.3 | IC50 | 3 | — | |
JXCFHCFAYKJVSI
|
7.3 | IC50 | 3 | — | |
RZJKWVPUWYLTJN
|
7.3 | IC50 | 3 | — | |
ADRJQPFHTSNURD
|
7.3 | IC50 | 2 | — | |
WEYWTPCHMFHABR
|
7.3 | Ki | 2 | — | |
ICSDSFFBTUMVKX
|
7.3 | Ki | 2 | — | |
DLMMMBXYCBMUDE
|
7.3 | IC50 | 2 | — | |
XRWGWRHXWJHKMY
|
7.2 | IC50 | 2 | — | |
XRWGWRHXWJHKMY
|
7.2 | IC50 | 2 | — | |
RYZQAFZHSBVEIT
|
7.2 | IC50 | 2 | — | |
KGOLFZSTQPOJBW
|
7.2 | IC50 | 2 | — | |
YJNWDJIIFRGLRO
|
7.2 | Ki | 6 | Yes | |
ITMQFUGUIZVZNR
|
7.1 | IC50 | 3 | — | |
KSLQUEKUGQKSAJ
|
7.1 | Ki | 4 | — | |
UHSLUGVLSJUOHH
|
7.1 | Ki | 3 | — | |
BVTSBOHKQXLEPE
|
7.1 | Ki | 2 | — | |
BXOTUFWBXZIMMA
|
7.1 | IC50 | 2 | — | |
FZURHBSSIFZNCU
|
7.1 | IC50 | 2 | — | |
DDYFSJLRMHFOPK
|
7.1 | IC50 | 2 | — | |
JXCFHCFAYKJVSI
|
7.1 | IC50 | 3 | — | |
RRWODDRPKAWHEH
|
7.1 | IC50 | 2 | — | |
LIOSIPYHSGHPQG
|
7.1 | Ki | 2 | — | |
AXQXSMSWAHKPFZ
|
7.0 | IC50 | 2 | — | |
UBQFBYMIHFXWBF
|
7.0 | IC50 | 3 | — | |
YSERSWXWBJFHEC
|
7.0 | IC50 | 2 | — | |
OLCPFVJJGLRGPS
|
7.0 | IC50 | 2 | — | |
JSAOPPSCSSMQLN
|
7.0 | IC50 | 2 | — | |
OYOZJKFWWAKHED
|
7.0 | IC50 | 3 | — | |
PRNNUULGNBSAAT
|
6.9 | IC50 | 2 | — | |
KWBQBHZSTYVPSB
|
6.9 | Ki | 3 | — | |
BZLKGVQCIONWMQ
|
6.9 | IC50 | 2 | — | |
LDLYNKUKWJPFHZ
|
6.9 | IC50 | 2 | — | |
LXTBWCJUTDGCHZ
|
6.9 | IC50 | 2 | — | |
DQYQHPUASSQDSB
|
6.9 | Ki | 3 | — | |
ITMFWUAKJPURIP
|
6.9 | Ki | 6 | Yes | |
KGOLFZSTQPOJBW
|
6.9 | IC50 | 2 | — | |
SSFFBSQJBLDEMQ
|
6.9 | IC50 | 2 | — | |
DQOBOCPZWNUNMH
|
6.8 | IC50 | 2 | — | |
DQZOBCXSUVKSEO
|
6.8 | IC50 | 2 | — |