Target Details
| UniProt AC | P08473 |
|---|---|
| Gene Symbol | MME |
| Protein Name | Neprilysin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01431 (Peptidase_M13) PF05649 (Peptidase_M13_N) |
Summary
- Multi-target molecules 252
- Clinical molecules 3
- Avg pChEMBL 7.77
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (252)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DOBNVUFHFMVMDB
|
8.2 | IC50 | 2 | — | |
RYAZPHMYWMQFFB
|
8.2 | Ki | 2 | — | |
XVXJQRXUEUIXNY
|
8.2 | Ki | 2 | — | |
AKSMLLXRBFIIDE
|
8.2 | IC50 | 2 | — | |
GKNJPJZPAMDYBU
|
8.2 | IC50 | 2 | — | |
PIBUIEXHVFJHNQ
|
8.2 | IC50 | 2 | — | |
LWRWHXRRIHLFGY
|
8.2 | IC50 | 2 | — | |
NWICWXQFBXWITN
|
8.2 | IC50 | 2 | — | |
ZGZOWIGWICXUAP
|
8.1 | IC50 | 2 | — | |
CERYYXRBRYOZMX
|
8.1 | IC50 | 2 | — | |
WSDIIIJALODSSH
|
8.1 | IC50 | 2 | — | |
YSERSWXWBJFHEC
|
8.1 | IC50 | 2 | — | |
UGLAENRVRPVULB
|
8.1 | IC50 | 2 | — | |
KSLGTDWGRDTBSU
|
8.1 | IC50 | 3 | — | |
OCDSLXZWNPDFJC
|
8.1 | IC50 | 3 | — | |
UOJKOYVPHFAXMP
|
8.1 | IC50 | 2 | — | |
HRBJATPCNVWLGP
|
8.0 | Ki | 3 | — | |
MKODWSWFPOSLLD
|
8.0 | IC50 | 2 | — | |
ASOTUXAPLNMLBP
|
7.9 | Ki | 2 | — | |
JRAQIPPUUOUHFM
|
7.9 | Ki | 2 | — | |
OJDOJGWVKJJLMB
|
7.9 | Ki | 3 | — | |
PRAUQXGSSFLOAP
|
7.9 | Ki | 3 | — | |
TYXFDFMUHPWCDX
|
7.8 | IC50 | 2 | — | |
ZVYGKCUEVQFXLW
|
7.8 | IC50 | 2 | — | |
FTZIHGUFMWZVIM
|
7.8 | IC50 | 3 | — | |
IMCHWZJWTLLCLS
|
7.8 | IC50 | 2 | — | |
QQKCLPWCRIGNMI
|
7.8 | IC50 | 2 | — | |
SYHXTELYVKDCHI
|
7.8 | IC50 | 2 | — | |
RZCHYBYQQJXXGU
|
7.7 | Ki | 3 | — | |
GSVWGGILYDYXLP
|
7.7 | IC50 | 2 | — | |
MAVHEVQROSUZGT
|
7.7 | IC50 | 3 | — | |
QQXJEPZLFZCIMX
|
7.7 | IC50 | 2 | — | |
HPLIOAAHFNYSEA
|
7.7 | IC50 | 2 | — | |
XLTCIQSQOMKREC
|
7.7 | IC50 | 2 | — | |
ISXNHFVFHVLVBQ
|
7.6 | Ki | 3 | — | |
YJSMEONIEBYZRH
|
7.6 | Ki | 3 | — | |
XBIYMMZPQYOOJC
|
7.6 | IC50 | 2 | — | |
SJZKJUPLQDZQPD
|
7.6 | IC50 | 3 | — | |
BKIADFDXLKFQRT
|
7.6 | Ki | 3 | — | |
BROFGMFOFNHCBY
|
7.6 | IC50 | 2 | — | |
DOBNVUFHFMVMDB
|
7.6 | IC50 | 2 | — | |
VSYYVORPLMQOJQ
|
7.5 | IC50 | 2 | — | |
ZPHBZEQOLSRPAK
|
7.5 | IC50 | 5 | — | |
PAQFIXCBKVQCFX
|
7.5 | IC50 | 2 | — | |
DPPTZNUVUSKYMF
|
7.5 | Ki | 4 | — | |
OSTXOFBATBEQSL
|
7.5 | IC50 | 3 | — | |
ZMFXEDLVSXEQSM
|
7.5 | IC50 | 3 | — | |
CRYGCPYTHSHCKP
|
7.5 | Ki | 2 | — | |
CZFGWEONSMKJRA
|
7.5 | Ki | 2 | — | |
HXSOGWMGAAJSIY
|
7.5 | Ki | 2 | — |