Target Details
| UniProt AC | P08473 |
|---|---|
| Gene Symbol | MME |
| Protein Name | Neprilysin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01431 (Peptidase_M13) PF05649 (Peptidase_M13_N) |
Summary
- Multi-target molecules 252
- Clinical molecules 3
- Avg pChEMBL 7.77
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (252)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PQBHIPADCOQVIZ
|
10.4 | IC50 | 2 | — | |
RIWRWPXUDHZKIO
|
10.1 | IC50 | 2 | — | |
SELXLNMHXRYMKY
|
9.7 | Ki | 2 | — | |
GNCWXHHRBZYERE
|
9.6 | Ki | 3 | — | |
MHSQCNUPGPCYGY
|
9.5 | IC50 | 2 | — | |
MYGUKWRMURCQGP
|
9.5 | IC50 | 2 | — | |
OFCQCSHBABYJSE
|
9.5 | IC50 | 2 | — | |
QLCPDIVEFVTPQJ
|
9.4 | IC50 | 2 | — | |
FHEAVMZMNOBKAV
|
9.4 | Ki | 2 | — | |
PMFRPUCBOVMLCM
|
9.3 | Ki | 2 | — | |
BLWJOUOTJGBSKF
|
9.2 | IC50 | 2 | — | |
DQULGQNMFILGNZ
|
9.2 | IC50 | 2 | — | |
VICZFKNTXNDQOA
|
9.2 | IC50 | 2 | — | |
BSJZYWSFNCKCDR
|
9.2 | IC50 | 3 | — | |
GFAPVUXBADBZKC
|
9.2 | IC50 | 2 | — | |
UQBKEHVOSNORFA
|
9.2 | Ki | 2 | — | |
XVTHDQIYTRAPLI
|
9.2 | IC50 | 2 | — | |
NAOAQOAPOBTFLY
|
9.1 | IC50 | 2 | — | |
HDIPKMHZRNJMPR
|
9.1 | Ki | 3 | — | |
MCEAHFJYQBFRCJ
|
9.1 | IC50 | 2 | — | |
UUMKQZVEZSXWBY
|
9.0 | IC50 | 2 | — | |
FAOLDJJTSITBOU
|
9.0 | IC50 | 2 | — | |
FPUIOUHUIOAZBC
|
9.0 | IC50 | 2 | — | |
NTLHWTOYJZOKBQ
|
9.0 | IC50 | 2 | — | |
ODIRGNPVJXPGMV
|
9.0 | IC50 | 2 | — | |
PUMGJIZLXLDCRQ
|
9.0 | IC50 | 2 | — | |
RPPNGIBDLYBJPM
|
9.0 | IC50 | 2 | — | |
ZJLMPQQUSAIJSM
|
9.0 | Ki | 2 | — | |
BNECOBGISSOLPT
|
9.0 | Ki | 3 | — | |
VNJDJPOTECLILR
|
8.9 | Ki | 2 | — | |
BBXMTNLJEHRMMT
|
8.9 | Ki | 3 | — | |
CDDHYPGPHOOMFW
|
8.9 | IC50 | 2 | — | |
CWJPVKSBGVPXRD
|
8.9 | Ki | 2 | — | |
BNECOBGISSOLPT
|
8.9 | Ki | 4 | — | |
LVRLSYPNFFBYCZ
|
8.9 | IC50 | 3 | — | |
WWTBZEKOSBFBEM
|
8.8 | Ki | 2 | — | |
RZMPSTCSWYMNIQ
|
8.8 | IC50 | 2 | — | |
ZBGYPMPWJWNWEA
|
8.8 | IC50 | 2 | — | |
OJCFZTVYDSKXNM
|
8.8 | Ki | 4 | — | |
OJCFZTVYDSKXNM
|
8.8 | Ki | 5 | — | |
QHBPFNHEJJZWMW
|
8.8 | IC50 | 2 | — | |
HTEXPDWHUAHOGC
|
8.7 | IC50 | 2 | — | |
IQHFJQXJLKTGJO
|
8.7 | IC50 | 2 | — | |
KSDXHWOIFKMBGX
|
8.7 | IC50 | 3 | — | |
NCJYNTULOJIUPY
|
8.7 | Ki | 2 | — | |
QXXMSEVVNUSHKJ
|
8.7 | Ki | 2 | — | |
QXXMSEVVNUSHKJ
|
8.7 | Ki | 2 | — | |
JQEZRNOCSSVLKH
|
8.7 | IC50 | 2 | — | |
GBKMVBCTZCVKSV
|
8.7 | IC50 | 2 | — | |
LPUDGHQMOAHMMF
|
8.7 | IC50 | 3 | — |