Target Details
| UniProt AC | P08311 |
|---|---|
| Gene Symbol | CTSG |
| Protein Name | Cathepsin G |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 85
- Clinical molecules 0
- Avg pChEMBL 7.31
KEGG Pathways (6)
Active Molecules (85)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FVFSUZHBTIUSFU
|
6.8 | Ki | 2 | — | |
HTMCLXGHJGHVGZ
|
6.8 | IC50 | 3 | — | |
BFPDTPAHEKIKHN
|
6.7 | IC50 | 2 | — | |
FVAHUQQSETWKRH
|
6.7 | Ki | 2 | — | |
NYGGGQOBPHOCIJ
|
6.7 | Ki | 3 | — | |
IMXJHAMVFYJETE
|
6.7 | IC50 | 2 | — | |
PDFLMEOJDBZIJL
|
6.6 | IC50 | 4 | — | |
WISJYGPAQGRLCK
|
6.6 | IC50 | 2 | — | |
PNILZVBINXNWHW
|
6.6 | Ki | 2 | — | |
VUEVZBHUKRORBJ
|
6.5 | IC50 | 2 | — | |
YDCSNPSSWBJJIR
|
6.5 | IC50 | 2 | — | |
BWTNDBKCQZCMSA
|
6.5 | IC50 | 2 | — | |
JBVRJKUPBUZDDJ
|
6.4 | Ki | 2 | — | |
GIHZBWSNGQZROH
|
6.4 | Ki | 2 | — | |
RMEUFAVEIHZTRM
|
6.4 | Ki | 4 | — | |
AQIIUWJCYOQHPS
|
6.4 | Ki | 2 | — | |
PJWRVDWTVAOOQV
|
6.3 | Ki | 7 | — | |
KTPYVEWDDQSBAX
|
6.3 | Ki | 5 | — | |
ZQSVKNYOSYOREJ
|
6.3 | Ki | 4 | — | |
GXJABQQUPOEUTA
|
6.2 | IC50 | 47 | — | |
JKRQSPIPAUZESC
|
6.2 | IC50 | 2 | — | |
NQXVELVXYLJZFV
|
6.2 | IC50 | 2 | — | |
VBQCUFXCAOKEJY
|
6.2 | Ki | 3 | — | |
PNEMWQVQIVXXIX
|
6.2 | IC50 | 2 | — | |
BIYZZFJCFHPBTP
|
6.2 | IC50 | 2 | — | |
FKSBHSQGFGGOEF
|
6.2 | Ki | 4 | — | |
GBDNHNNAGDSWAW
|
6.2 | Ki | 4 | — | |
LFIXADISWCDQHZ
|
6.2 | Ki | 4 | — | |
QQBRBPSSMDPLLA
|
6.1 | Ki | 5 | — | |
YGRSMPVCBHOYMS
|
6.1 | Ki | 2 | — | |
BYVVCQVQZLFQOJ
|
6.1 | IC50 | 3 | — | |
YVERQXIEPUPSEH
|
6.1 | IC50 | 2 | — | |
VUWARVVMIAAMOY
|
6.0 | IC50 | 3 | — | |
GKBXJOCPZBRUIG
|
6.0 | IC50 | 4 | — | |
AEVPIESDIOSSSM
|
6.0 | IC50 | 2 | — |